SCHEMBL6025944

SCHEMBL6025944

ClC(OCc1ccccc1)OC(Cl)OCc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.48
IDO1 P14902 1/20 0.44
SLC1A3 P43003 2/20 0.43
SLC1A2 P43004 2/20 0.43
SLC1A1 P43005 2/20 0.43
CYP1A2 P05177 2/20 0.43
CYP2C19 P33261 2/20 0.43
MEN1 O00255 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
KMT2A Q03164 1/20 0.43
AGXT P21549 1/20 0.43
ALDH1A1 P00352 2/20 0.42
SLC6A2 P23975 3/20 0.41
SLC6A3 Q01959 3/20 0.41
SLC6A4 P31645 2/20 0.41
CHRNB2 P17787 1/20 0.41
CHRNA4 P43681 1/20 0.41
CA1 P00915 3/20 0.38
CA2 P00918 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL71045 0.83 TSHR (0.44) TSHRIDO1SLC1A3SLC1A2SLC1A1
SCHEMBL10344292 0.81 TSHR (0.52) TSHRIDO1SLC1A3SLC1A2SLC1A1
SCHEMBL3292550 0.81 TSHR (0.43) TSHRIDO1SLC1A3SLC1A2SLC1A1
SCHEMBL5503634 0.77 TSHR (0.48) TSHRIDO1SLC1A3SLC1A2SLC1A1
SCHEMBL7302690 0.77 TSHR (0.48) TSHRIDO1SLC1A3SLC1A2SLC1A1
SCHEMBL7302683 0.77 TSHR (0.48) TSHRIDO1SLC1A3SLC1A2SLC1A1
SCHEMBL8079929 0.76 TSHR (0.52) TSHRIDO1SLC1A3SLC1A2SLC1A1
SCHEMBL547986 0.76 SLC6A2 (0.47) TSHRIDO1SLC1A3SLC1A2SLC1A1
SCHEMBL14667806 0.76 TSHR (0.46) TSHRIDO1SLC1A3SLC1A2SLC1A1
SCHEMBL6774650 0.75 TSHR (0.57) TSHRIDO1SLC1A3SLC1A2SLC1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107383139-A The method that a kind of β cholanic acid new derivatives of 7 oxo of 3 α hydroxyls 5 prepare shellfish cholic acid difficult to understand 杭州和泽医药科技有限公司 2017-11-24 CN disclosed
CN-103450113-B Thiadiazine-triketones-substituted derivative, preparation method thereof and application UNIV SHANDONG 2014-12-10 CN disclosed
CN-103450113-A Thiadiazine-triketones-substituted derivative, preparation method thereof and application UNIV SHANDONG 2013-12-18 CN disclosed
EP-1369490-B1 Method of preparing a composition containing hygromycin A and epi-hygromycin PFIZER PROD INC (US) 2006-02-08 EP disclosed
EP-1369490-A1 Method of preparing a composition containing hygromycin A and epi-hygromycin Pfizer Products Inc. (US) 2003-12-10 EP disclosed
EP-1075483-B1 HYGROMYCIN A DERIVATIVES PFIZER PROD INC (US) 2003-12-03 EP disclosed
US-6313100-B1 ANTIBACTERIAL, ANTIPROTOZOA AGENTS PFIZER INC 2001-11-06 US disclosed
EP-1075483-A2 HYGROMYCIN A DERIVATIVES Pfizer Products Inc. (US) 2001-02-14 EP disclosed
WO-1999057125-A2 HYGROMYCIN A DERIVATIVES PFIZER PRODUCTS INC. (US) 1999-11-11 WO disclosed
US-5760018-A Gem-disubstituted azacyclic tachykinin antagonists MERCK SHARP & DOHME LTD. (GB) 1998-06-02 US disclosed
EP-0739336-A1 GEM-DISUBSTITUTED AZACYCLIC TACHYKININ ANTAGONISTS MERCK SHARP & DOHME LTD. (GB) 1996-10-30 EP disclosed
WO-1995028413-A1 17β-SUBSTITUTED 3-CARBOXY STEROIDS THAT INHIBIT 5-α-REDUCTASE SMITHKLINE BEECHAM CORPORATION (US) 1995-10-26 WO disclosed
WO-1995019344-A1 GEM-DISUBSTITUTED AZACYCLIC TACHYKININ ANTAGONISTS MERCK SHARP & DOHME LIMITED (GB) 1995-07-20 WO disclosed