SCHEMBL547986

SCHEMBL547986

ClC(OCc1ccccc1)c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 3/20 0.47
SLC6A4 P31645 3/20 0.47
SLC6A3 Q01959 3/20 0.47
CHRNB2 P17787 1/20 0.47
CHRNA4 P43681 1/20 0.47
TSHR P16473 2/20 0.46
TACR1 P25103 2/20 0.43
IDO1 P14902 1/20 0.43
SLC1A3 P43003 2/20 0.42
SLC1A2 P43004 2/20 0.42
SLC1A1 P43005 2/20 0.42
MEN1 O00255 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
KMT2A Q03164 1/20 0.42
AGXT P21549 1/20 0.41
ALDH1A1 P00352 1/20 0.41
AOC3 Q16853 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6181884 0.88 CHRNB2 (0.63) SLC6A2SLC6A4SLC6A3CHRNB2CHRNA4
SCHEMBL28534097 0.87 CHRNB2 (0.45) SLC6A2SLC6A4SLC6A3CHRNB2CHRNA4
SCHEMBL28528002 0.87 CHRNB2 (0.45) SLC6A2SLC6A4SLC6A3CHRNB2CHRNA4
SCHEMBL28531540 0.87 CHRNB2 (0.45) SLC6A2SLC6A4SLC6A3CHRNB2CHRNA4
SCHEMBL4599464 0.82 IDO1 (0.45) SLC6A2SLC6A4SLC6A3CHRNB2CHRNA4
SCHEMBL28531048 0.80 EPHX1 (0.47) SLC6A4CHRNB2CHRNA4TSHRALDH1A1
SCHEMBL10344292 0.79 TSHR (0.52) SLC6A2SLC6A4SLC6A3CHRNB2CHRNA4
SCHEMBL11100946 0.77 SLC6A2 (0.50) SLC6A2SLC6A4SLC6A3CHRNB2CHRNA4
SCHEMBL10431978 0.77 SLC6A2 (0.50) SLC6A2SLC6A4SLC6A3CHRNB2CHRNA4
SCHEMBL29277741 0.77 SLC6A2 (0.50) SLC6A2SLC6A4SLC6A3CHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 72 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0873293-B1 IMPROVED PROCESS FOR THE PREPARATION OF ALKYL OR ARYL ALDEHYDE INTERMEDIATES ABBOTT LAB (US) 2001-07-25 EP claimed
EP-0873293-A1 IMPROVED PROCESS FOR THE PREPARATION OF ALKYL OR ARYL ALDEHYDE INTERMEDIATES Abbott Laboratories (US) 1998-10-28 EP claimed
WO-1997023439-A1 IMPROVED PROCESS FOR THE PREPARATION OF ALKYL OR ARYL ALDEHYDE INTERMEDIATES ABBOTT LABORATORIES (US) 1997-07-03 WO claimed
EP-3030555-B1 NOVEL PYRAZINE AMIDE COMPOUNDS BOEHRINGER INGELHEIM INT (DE) 2019-01-30 EP disclosed
CN-106349105-B A kind of preparation method of benzyl cyanide 河北诚信集团有限公司 2018-11-27 CN disclosed
EP-2470512-B1 AROMATASE INHIBITOR ESTRYX PHARMA LTD (GB) 2018-05-02 EP disclosed
CN-104530047-B Ketone quaternary ammonium salt of iron dung rice 6 and preparation method and application 西北农林科技大学 2017-11-10 CN disclosed
CN-106349105-A Preparation method of substituted benzyl cyanide 河北诚信有限责任公司 2017-01-25 CN disclosed
EP-3030555-A1 NOVEL PYRAZINE AMIDE COMPOUNDS Boehringer Ingelheim International GmbH (DE) 2016-06-15 EP disclosed
CN-102596919-B Aromatase inhibitor STRIX LTD. (GB) 2015-11-25 CN disclosed
US-9096548-B2 Pyrazine amide compounds BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2015-08-04 US disclosed
US-5401851-A Preparation of proline derivatives ELI LILLY AND COMPANY (US) 1995-03-28 US disclosed
CN-1098714-A The 1H-indole-3-acetic acid hydrazide spla 2 inhibitors LILLY CO ELI (US) 1995-02-15 CN disclosed
CN-1085897-A Angiotension II antagonists LILLY CO ELI (US) 1994-04-27 CN disclosed
EP-0573271-A1 Angiotensin II antagonists ELI LILLY AND COMPANY (US) 1993-12-08 EP disclosed
EP-0565317-A1 (2-(2-hydroxy-2 phenylethylamino)ethoxy) phenyl derivatives, processes and intermediates for their preparation, pharmaceutical compositions containing them and their use as Beta-3-adrenoceptor agonists ZENECA LIMITED (GB) 1993-10-13 EP disclosed
WO-1993000359-A1 MODIFIED PEPTIDES TRANSPORTABLE INTO THE CENTRAL NERVOUS SYSTEM THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1993-01-07 WO disclosed
EP-0183216-B1 N-(ARALKOXYBENZYL)-4(BENZHYDRYL) PIPERIDINES G.D. Searle & Co. (US) 1989-07-19 EP disclosed
US-4650874-A CARDIOVASCULAR AGENTS G. D. SEARLE & CO. (US) 1987-03-17 US disclosed
EP-0183216-A1 N-(Aralkoxybenzyl)-4(benzhydryl) piperidines G.D. Searle & Co. (US) 1986-06-04 EP disclosed