SCHEMBL6026299

SCHEMBL6026299

CCOC(=O)c1nc(C)n(C2CC2)c1C.Cc1nc(CO)c(C)n1C1CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRK6 P43250 1/20 0.39
CNR2 P34972 1/20 0.38
OGFRL1 Q5TC84 4/20 0.37
OPRM1 P35372 3/20 0.37
OPRK1 P41145 3/20 0.37
OPRD1 P41143 2/20 0.37
ALDH1A1 P00352 3/20 0.36
KDM4E B2RXH2 1/20 0.36
HPGD P15428 1/20 0.36
CYP1A2 P05177 1/20 0.36
KMT2A Q03164 1/20 0.36
TP53 P04637 1/20 0.35
ALOX12 P18054 1/20 0.35
ELANE P08246 1/20 0.35
RCE1 Q9Y256 1/20 0.35
GAA P10253 1/20 0.34
TSHR P16473 1/20 0.34
HTT P42858 1/20 0.34
HSD17B10 Q99714 1/20 0.34
USP2 O75604 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5038584 0.91 GRK6 (0.44) GRK6CNR2OGFRL1OPRM1OPRK1
SCHEMBL2681871 0.85 CNR2 (0.50) GRK6CNR2OGFRL1OPRM1OPRK1
SCHEMBL5048090 0.82 CNR2 (0.34) CNR2ALDH1A1KDM4EKMT2AGAA
SCHEMBL6026302 0.73 GRK6 (0.33) GRK6CNR2OGFRL1OPRM1OPRK1
SCHEMBL4734637 0.71 CNR2 (0.48) CNR2OGFRL1OPRM1OPRK1OPRD1
SCHEMBL14886782 0.68 HPGD (0.38) ALDH1A1KDM4EHPGDCYP1A2KMT2A
SCHEMBL12926023 0.68 KMT2A (0.46) ALDH1A1KDM4EHPGDCYP1A2KMT2A
SCHEMBL16268486 0.68 GRK6 (0.42) GRK6OGFRL1OPRM1OPRK1OPRD1
SCHEMBL30668018 0.66 GRK6 (0.43) GRK6OGFRL1OPRM1OPRK1OPRD1
SCHEMBL20386876 0.64 KMT2A (0.43) ALDH1A1CYP1A2KMT2ATP53ALOX12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1644351-A1 IMIDAZOLE DERIVATIVES III F. HOFFMANN-LA ROCHE AG (CH) 2006-04-12 EP disclosed
WO-2005003117-A1 IMIDAZOLE DERIVATIVES III F. HOFFMANN-LA ROCHE AG (CH) 2005-01-13 WO disclosed