SCHEMBL6028857

SCHEMBL6028857

COc1ccc(C2CCOCC2)c2sc(NC(=O)N(C)C3CCC(C)(O)CC3)nc12

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 15/20 0.49
ADORA1 P30542 13/20 0.49
ADORA2B P29275 4/20 0.49
ADORA3 P0DMS8 1/20 0.49
ALDH1A1 P00352 3/20 0.45
MAPT P10636 1/20 0.45
TSHR P16473 1/20 0.45
HSD17B10 Q99714 1/20 0.45
KDM4E B2RXH2 2/20 0.41
HPGD P15428 2/20 0.41
PKM P14618 1/20 0.40
ATM Q13315 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CHRM4 P08173 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5040964 1.00 ADORA2A (0.49) ADORA2AADORA1ADORA2BADORA3ALDH1A1
SCHEMBL5036082 0.92 ALDH1A1 (0.51) ADORA2AADORA1ADORA2BADORA3ALDH1A1
SCHEMBL5035824 0.90 ADORA2A (0.50) ADORA2AADORA1ADORA2BADORA3ALDH1A1
SCHEMBL5035822 0.90 ADORA2A (0.50) ADORA2AADORA1ADORA2BADORA3ALDH1A1
SCHEMBL5039395 0.90 ADORA2A (0.50) ADORA2AADORA1ADORA2BADORA3ALDH1A1
SCHEMBL5133408 0.88 ALDH1A1 (0.48) ADORA2AADORA1ADORA2BADORA3ALDH1A1
SCHEMBL5040911 0.87 ADORA2A (0.47) ADORA2AADORA1ADORA2BADORA3ALDH1A1
SCHEMBL5039672 0.87 ADORA2A (0.47) ADORA2AADORA1ADORA2BADORA3ALDH1A1
SCHEMBL5561806 0.87 ADORA2A (0.45) ADORA2AADORA1ADORA2BADORA3ALDH1A1
SCHEMBL5561811 0.87 ADORA2A (0.45) ADORA2AADORA1ADORA2BADORA3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1636223-A1 BENZOTHIAZOLE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS F. Hoffman-la Roche AG (CH) 2006-03-22 EP disclosed
WO-2005000842-A1 BENZOTHIAZOLE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS F. HOFFMAN-LA ROCHE AG (CH) 2005-01-06 WO disclosed