SCHEMBL6032269

SCHEMBL6032269

COc1c2c(c(Br)[nH]c1=O)CCN(Cc1ccc(F)c(Cl)c1)C2=O.COc1c2c(c(Br)[nH]c1=O)CCN(Cc1ccc(F)c(Cl)c1)C2=O

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 5/20 0.37
DAO P14920 1/20 0.37
EZH2 Q15910 9/20 0.37
HTR2A P28223 1/20 0.37
GRM2 Q14416 1/20 0.37
TNIK Q9UKE5 1/20 0.35
GAA P10253 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4486283 1.00 P2RX7 (0.37) P2RX7DAOEZH2HTR2AGRM2
SCHEMBL4478453 0.86 DAO (0.39) DAOEZH2HTR2AGRM2TNIK
SCHEMBL1336948 0.86 AKR1B1 (0.38) P2RX7DAOEZH2HTR2AGRM2
SCHEMBL4492829 0.84 AKR1B1 (0.35) P2RX7DAOEZH2HTR2AGRM2
SCHEMBL4484368 0.83 MEN1 (0.39) EZH2ALDH1A1LMNAHTTSMN1; SMN2
SCHEMBL4482140 0.83 P2RX7 (0.39) P2RX7EZH2HTR2AGRM2ALDH1A1
SCHEMBL4486261 0.78 P2RX7 (0.37) P2RX7EZH2HTR2AGRM2ALDH1A1
SCHEMBL4479378 0.77 EZH2 (0.37) P2RX7EZH2HTR2AGRM2ALDH1A1
SCHEMBL3023303 0.77 EZH2 (0.32) EZH2HTR2AGRM2
SCHEMBL1336823 0.77 EZH2 (0.32) EZH2HTR2AGRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1725556-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2006-11-29 EP disclosed
WO-2005087768-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 2005-09-22 WO disclosed