SCHEMBL6033076

SCHEMBL6033076

FC(F)(F)c1ccc(Nc2cc(-c3ccc4cccnc4c3)ncn2)cn1.FC(F)(F)c1ccc(Nc2cc(-c3ccc4cccnc4c3)ncn2)nc1

nearest known ligand 0.67

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 12/20 0.67
ABL1 P00519 4/20 0.56
BCR P11274 4/20 0.56
TNNI3K Q59H18 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5801083 0.92 TRPV1 (0.69) TRPV1ABL1BCR
SCHEMBL5797628 0.91 TRPV1 (0.70) TRPV1ABL1BCRTNNI3K
SCHEMBL4832759 0.85 TRPV1 (0.87) TRPV1ABL1BCRTNNI3K
SCHEMBL6252940 0.84 TRPV1 (0.65) TRPV1ABL1BCRTNNI3K
SCHEMBL6033561 0.81 TRPV1 (0.61) TRPV1
SCHEMBL13868105 0.81 TRPV1 (1.00) TRPV1ABL1BCR
SCHEMBL4837497 0.77 TRPV1 (0.76) TRPV1ABL1BCRTNNI3K
SCHEMBL1011253 0.74 TRPV1 (0.83) TRPV1ABL1BCR
SCHEMBL4832960 0.73 ABL1 (0.72) TRPV1ABL1BCRTNNI3K
SCHEMBL12943132 0.73 ABL1 (1.00) TRPV1ABL1BCR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1685124-A1 SUBSTITUTED NITROGEN-CONTAINING SIX-MEMBERED AMINO-HETEROCYCLES AS VANILLOID-1 RECEPTOR ANTAGONISTS FOR TREATING PAIN MERCK SHARP & DOHME LTD. (GB) 2006-08-02 EP disclosed
WO-2005047279-A1 SUBSTITUTED NITROGEN-CONTAINING SIX-MEMBERED AMINO-HETEROCYCLES AS VANILLOID-1 RECEPTOR ANTAGONISTS FOR TREATING PAIN MERCK SHARP & DOHME LIMITED (GB) 2005-05-26 WO disclosed