SCHEMBL6037055

SCHEMBL6037055

CC(/C=C/CC1CCc2cc3c(cc21)C(C)(C)CCC3(C)C)=C\C(=O)O

nearest known ligand 0.52

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
RXRA P19793 20/20 0.52
RXRG P48443 15/20 0.52
RARG P13631 7/20 0.50
RARB P10826 7/20 0.50
RARA P10276 3/20 0.50
RXRB P28702 13/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6037057 1.00 RXRA (0.52) RXRARXRGRARGRARBRARA
SCHEMBL6037042 0.94 RXRA (0.52) RXRARXRGRARGRARBRARA
SCHEMBL6037041 0.94 RXRA (0.52) RXRARXRGRARGRARBRARA
SCHEMBL8309204 0.81 RXRA (0.48) RXRARXRGRARGRARBRARA
SCHEMBL8309207 0.81 RXRA (0.48) RXRARXRGRARGRARBRARA
SCHEMBL6037059 0.71 RXRA (0.53) RXRARXRGRARGRARBRARA
SCHEMBL6037060 0.71 RXRA (0.53) RXRARXRGRARGRARBRARA
SCHEMBL6037045 0.71 RXRA (0.52) RXRARXRGRARGRARBRARA
SCHEMBL6037047 0.71 RXRA (0.52) RXRARXRGRARGRARBRARA
SCHEMBL6037058 0.70 RXRA (0.52) RXRARXRGRARGRARBRARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0933350-A1 Tricyclic retinoids, methods for their production and use LIGAND PHARMACEUTICALS INCORPORATED (US) 1999-08-04 EP claimed
EP-0800504-A1 TRICYCLIC RETINOIDS, METHODS FOR THEIR PRODUCTION AND USE LIGAND PHARMACEUTICALS, INC. (US) 1997-10-15 EP claimed
WO-1996020914-A1 TRICYCLIC RETINOIDS, METHODS FOR THEIR PRODUCTION AND USE LIGAND PHARMACEUTICALS INCORPORATED (US) 1996-07-11 WO claimed
US-20060030597-A1 Method of inhibiting angiogenesis GERRITSEN MARY E 2006-02-09 US disclosed
US-20010036955-A1 Method of inhibiting angiogenesis GENENTECH, INC. 2001-11-01 US disclosed
EP-0933351-A1 Tricyclic retinoids, methods for their production and use LIGAND PHARMACEUTICALS INCORPORATED (US) 1999-08-04 EP disclosed
EP-0933350-A1 Tricyclic retinoids, methods for their production and use LIGAND PHARMACEUTICALS INCORPORATED (US) 1999-08-04 EP disclosed
EP-0800504-A1 TRICYCLIC RETINOIDS, METHODS FOR THEIR PRODUCTION AND USE LIGAND PHARMACEUTICALS, INC. (US) 1997-10-15 EP disclosed
WO-1996020914-A1 TRICYCLIC RETINOIDS, METHODS FOR THEIR PRODUCTION AND USE LIGAND PHARMACEUTICALS INCORPORATED (US) 1996-07-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060030597-A1 Method of inhibiting angiogenesis PPARG, PPARA, RXRG RXRA 6/4885RXRG 3/4885RARG 10/4885
US-20010036955-A1 Method of inhibiting angiogenesis PPARG, PPARA, RXRG RXRA 6/4885RXRG 3/4885RARG 10/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.