SCHEMBL6046381

SCHEMBL6046381

CC(Cc1cccc(C(=O)NCC(C)(C)c2ccc(O)cc2)c1)NCC(O)c1ccc(O)c(NC=O)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 16/20 0.53
ADRB1 P08588 6/20 0.53
ADRB3 P13945 4/20 0.53
DRD2 P14416 2/20 0.53
CYP1A2 P05177 2/20 0.53
CYP3A4 P08684 2/20 0.53
CYP2D6 P10635 2/20 0.53
TSHR P16473 2/20 0.53
MAPK1 P28482 2/20 0.53
PGR P06401 1/20 0.53
SLC6A4 P31645 1/20 0.53
ADRA1A P35348 1/20 0.53
PTGS2 P35354 1/20 0.53
SLC6A3 Q01959 1/20 0.53
CYP2C19 P33261 1/20 0.53
DRD3 P35462 1/20 0.53
CASP3 P42574 1/20 0.49
CASP6 P55212 1/20 0.49
NFKB1 P19838 1/20 0.44
RAB9A P51151 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3627693 1.00 ADRB2 (0.53) ADRB2ADRB1ADRB3DRD2CYP1A2
SCHEMBL3626078 1.00 ADRB2 (0.53) ADRB2ADRB1ADRB3DRD2CYP1A2
SCHEMBL3626067 1.00 ADRB2 (0.53) ADRB2ADRB1ADRB3DRD2CYP1A2
SCHEMBL3627697 1.00 ADRB2 (0.53) ADRB2ADRB1ADRB3DRD2CYP1A2
SCHEMBL3619508 0.87 ADRB2 (0.41) ADRB2ADRB1ADRB3DRD2CYP1A2
SCHEMBL5584105 0.87 ADRB2 (0.41) ADRB2ADRB1ADRB3DRD2CYP1A2
SCHEMBL3619519 0.87 ADRB2 (0.41) ADRB2ADRB1ADRB3DRD2CYP1A2
SCHEMBL3625042 0.87 ADRB2 (0.50) ADRB2ADRB1
SCHEMBL3625038 0.87 ADRB2 (0.50) ADRB2ADRB1
SCHEMBL4430362 0.79 ADRB2 (0.80) ADRB2ADRB1ADRB3DRD2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730103-A1 FORMAMIDE DERIVATIVES USEFUL AS ADRENOCEPTOR Pfizer Limited (GB) 2006-12-13 EP disclosed
WO-2005092840-A1 FORMAMIDE DERIVATIVES USEFUL AS ADRENOCEPTOR PFIZER LIMITED (GB) 2005-10-06 WO disclosed