SCHEMBL6053607

SCHEMBL6053607

COc1ccccc1N1CCN(CCCCNC(=O)c2ccc(Cl)cc2)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 16/20 0.94
DRD3 P35462 16/20 0.94
DRD4 P21917 9/20 0.93
HTR1A P08908 2/20 0.83
ADRA1D P25100 1/20 0.83
ADRA1A P35348 1/20 0.83
ADRA1B P35368 1/20 0.83
KCNH2 Q12809 1/20 0.81
CYP1A2 P05177 1/20 0.79
MAPT P10636 1/20 0.79
CYP2C9 P11712 1/20 0.79
CYP2C19 P33261 1/20 0.79
SMN1; SMN2 Q16637 1/20 0.79

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14761722 0.92 DRD2 (1.00) DRD2DRD3DRD4HTR1AADRA1D
SCHEMBL14761605 0.91 DRD2 (0.98) DRD2DRD3DRD4HTR1AADRA1D
SCHEMBL10950772 0.90 DRD2 (0.98) DRD2DRD3DRD4HTR1AADRA1D
SCHEMBL17194866 0.90 DRD2 (1.00) DRD2DRD3DRD4HTR1AADRA1D
SCHEMBL14005958 0.89 DRD2 (0.79) DRD2DRD3DRD4HTR1AADRA1D
SCHEMBL14761584 0.88 DRD2 (0.94) DRD2DRD3DRD4HTR1AADRA1D
SCHEMBL27978158 0.88 DRD2 (1.00) DRD2DRD3DRD4HTR1AADRA1D
SCHEMBL1156684 0.88 DRD2 (1.00) DRD2DRD3DRD4HTR1AADRA1D
SCHEMBL10910646 0.88 DRD2 (0.94) DRD2DRD3DRD4HTR1AADRA1D
SCHEMBL9653369 0.86 DRD3 (0.72) DRD2DRD3DRD4HTR1AADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1272223-B1 THERAPEUTIC AND DIAGNOSTIC LIGAND SYSTEMS COMPRISING TRANSPORT MOLECULE BINDING PROPERTIES AND MEDICAMENTS CONTAINING THE SAME KTB TUMORFORSCHUNGS GMBH (DE) 2006-05-31 EP disclosed