SCHEMBL6054147

SCHEMBL6054147

C[C@H](NC1(c2ccccc2C(C)(C)C)CCCCO1)C(=O)N[C@H](C=O)CC(=O)O

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 15/20 0.37
CASP3 P42574 2/20 0.33
CASP6 P55212 1/20 0.33
CASP8 Q14790 1/20 0.33
IL1B P01584 1/20 0.33
CTSL P07711 2/20 0.33
CTSB P07858 2/20 0.33
CTSK P43235 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6054164 0.92 HDAC4 (0.37) CASP1IL1BCTSK
SCHEMBL5669625 0.92 CASP1 (0.39) CASP1CASP3CASP6CASP8
SCHEMBL6054175 0.87 CASP1 (0.38) CASP1CASP3IL1BCTSLCTSB
SCHEMBL6054163 0.87 CASP1 (0.38) CASP1CASP3IL1BCTSLCTSB
SCHEMBL6054155 0.87 PTGS1 (0.32) CASP1CASP3IL1B
SCHEMBL6054149 0.86 CASP1 (0.39) CASP1CASP3CASP6CASP8IL1B
SCHEMBL6054185 0.86 CASP1 (0.45) CASP1CASP3
SCHEMBL6054158 0.85 CASP1 (0.39) CASP1CASP3IL1BCTSLCTSB
SCHEMBL1896165 0.84 CASP1 (0.38) CASP1CASP3CASP6CASP8
SCHEMBL6054181 0.82 CASP1 (0.37) CASP1IL1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7053056-B2 C-terminal modified oxamyl dipeptides as inhibitors of the ICE/ced-3 family of cysteine proteases IDUN PHARMACEUTICALS, INC. (US) 2006-05-30 US claimed