SCHEMBL6054249

SCHEMBL6054249

CCOC(=O)c1cn2ncc(C#N)c(N3CCNCC3)c2c1C

nearest known ligand 0.55

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAP2K1 Q02750 12/20 0.55
ALDH1A1 P00352 2/20 0.50
RET P07949 4/20 0.47
KDM4E B2RXH2 2/20 0.42
POLB P06746 1/20 0.42
HTT P42858 1/20 0.42
RECQL P46063 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6054312 0.87 MAP2K1 (0.55) MAP2K1ALDH1A1RETKDM4EPOLB
SCHEMBL6054378 0.85 MAP2K1 (0.53) MAP2K1RETKDM4EPOLBHTT
SCHEMBL6054328 0.83 RET (0.54) MAP2K1RET
SCHEMBL6054224 0.82 MAP2K1 (0.58) MAP2K1ALDH1A1RETKDM4EPOLB
SCHEMBL6054246 0.82 MAP2K1 (0.59) MAP2K1ALDH1A1RETKDM4E
SCHEMBL6054292 0.79 MAP2K1 (0.61) MAP2K1ALDH1A1KDM4EPOLBHTT
SCHEMBL3687662 0.79 MAP2K1 (0.63) MAP2K1ALDH1A1KDM4EPOLBHTT
SCHEMBL3692161 0.73 MAP2K1 (0.96) MAP2K1ALDH1A1KDM4EHTT
SCHEMBL3690032 0.73 MAP2K1 (0.62) MAP2K1KDM4EPOLBHTTRECQL
SCHEMBL6054273 0.72 MAP2K1 (0.61) MAP2K1KDM4EPOLBHTTRECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7030112-B2 Pyrrolopyridazine compounds and methods of use thereof for the treatment of proliferative disorders BRISTOL-MYERS SQUIBB COMPANY (US) 2006-04-18 US claimed
US-7030112-B2 Pyrrolopyridazine compounds and methods of use thereof for the treatment of proliferative disorders BRISTOL-MYERS SQUIBB COMPANY (US) 2006-04-18 US disclosed