SCHEMBL6054292

SCHEMBL6054292

CCOC(=O)c1cn2ncc(C#N)c(NC3CCNCC3)c2c1C

nearest known ligand 0.61

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MAP2K1 Q02750 14/20 0.61
ALDH1A1 P00352 2/20 0.43
KDM4E B2RXH2 2/20 0.42
POLB P06746 1/20 0.42
HTT P42858 1/20 0.42
RECQL P46063 1/20 0.42
PDE4B Q07343 2/20 0.40
PLAT P00750 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3690032 0.91 MAP2K1 (0.62) MAP2K1KDM4EPOLBHTTRECQL
SCHEMBL6054273 0.90 MAP2K1 (0.61) MAP2K1KDM4EPOLBHTTRECQL
SCHEMBL6054279 0.87 MAP2K1 (0.59) MAP2K1KDM4EPOLBHTTRECQL
SCHEMBL6054304 0.84 MAP2K1 (0.55) MAP2K1ALDH1A1
SCHEMBL6054389 0.83 MAP2K1 (0.64) MAP2K1ALDH1A1KDM4E
SCHEMBL6054249 0.79 MAP2K1 (0.55) MAP2K1ALDH1A1KDM4EPOLBHTT
SCHEMBL6054224 0.77 MAP2K1 (0.58) MAP2K1ALDH1A1KDM4EPOLBHTT
SCHEMBL5801667 0.77 MAP2K1 (0.56) MAP2K1
SCHEMBL3687662 0.76 MAP2K1 (0.63) MAP2K1ALDH1A1KDM4EPOLBHTT
SCHEMBL5137524 0.76 MAP2K1 (0.55) MAP2K1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7030112-B2 Pyrrolopyridazine compounds and methods of use thereof for the treatment of proliferative disorders BRISTOL-MYERS SQUIBB COMPANY (US) 2006-04-18 US claimed
US-7030112-B2 Pyrrolopyridazine compounds and methods of use thereof for the treatment of proliferative disorders BRISTOL-MYERS SQUIBB COMPANY (US) 2006-04-18 US disclosed