SCHEMBL6056590

SCHEMBL6056590

CC(C)(C)Oc1ccc(C(F)(F)F)cc1CC(O)CNC(=O)C1CCC(=O)C1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.39
KMT2A Q03164 3/20 0.37
SCN9A Q15858 3/20 0.35
EPHX2 P34913 2/20 0.35
SSTR4 P31391 1/20 0.34
SCN1A P35498 1/20 0.33
SCN5A Q14524 1/20 0.33
XIAP P98170 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
PPARD Q03181 1/20 0.32
PPARA Q07869 1/20 0.32
ADAMTS4 O75173 2/20 0.32
MMP2 P08253 2/20 0.32
MMP3 P08254 2/20 0.32
MMP12 P39900 2/20 0.32
MMP13 P45452 2/20 0.32
MMP14 P50281 2/20 0.32
ADAMTS5 Q9UNA0 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6056589 0.74 PTGDR2 (0.44) SCN9APTGDR2
SCHEMBL6056617 0.70 EPHX2 (0.41) POLBKMT2AEPHX2SSTR4PPARD
SCHEMBL3165046 0.66 PPARD (0.38) PPARDPPARA
SCHEMBL5729938 0.66 CCR2 (0.49) POLBKMT2ANPC1RAB9A
SCHEMBL14169388 0.65 EPHX2 (0.40) POLBKMT2AEPHX2SSTR4PTGDR2
SCHEMBL3170727 0.65 CCR2 (0.42) PPARDPPARA
SCHEMBL3164000 0.64 CCR2 (0.41) PPARDPPARA
SCHEMBL2637443 0.61 IDO1 (0.41) SCN9ARAB9A
SCHEMBL14513598 0.61 CCR2 (0.52)
SCHEMBL3623332 0.61 PPARD (0.38) PTGDR2PPARDPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1615699-A2 BENZOXAZINYL-AMIDOCYCLOPENTYL-HETEROCYCLIC MODULATORS OF CHEMOKINE RECEPTORS Merck & Co., Inc. (US) 2006-01-18 EP disclosed
WO-2004092124-A2 BENZOXAZINYL-AMIDOCYCLOPENTYL-HETEROCYCLIC MODULATORS OF CHEMOKINE RECEPTORS MERCK & CO., INC. (US) 2004-10-28 WO disclosed