SCHEMBL6058660

SCHEMBL6058660

CC(C)(C)OC(=O)N[C@H]1C=C[C@@H](CBr)C1

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NFKB1 P19838 6/20 0.54
NFKB2 Q00653 6/20 0.54
RELA Q04206 6/20 0.54
KDM1A O60341 2/20 0.39
BTK Q06187 1/20 0.39
KMT2A Q03164 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
GAA P10253 1/20 0.38
MAOB P27338 2/20 0.38
MAOA P21397 1/20 0.38
EPHX2 P34913 1/20 0.37
AKT1 P31749 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6058662 1.00 NFKB1 (0.54) NFKB1NFKB2RELAKDM1ABTK
SCHEMBL6058659 1.00 NFKB1 (0.54) NFKB1NFKB2RELAKDM1ABTK
SCHEMBL3906310 0.86 NFKB1 (0.51) NFKB1NFKB2RELAKDM1ABTK
SCHEMBL31454839 0.86 NFKB1 (0.51) NFKB1NFKB2RELAKDM1ABTK
SCHEMBL31454797 0.86 NFKB1 (0.51) NFKB1NFKB2RELAKDM1ABTK
SCHEMBL4998586 0.86 NFKB1 (0.51) NFKB1NFKB2RELAKDM1ABTK
SCHEMBL5016759 0.86 NFKB1 (0.51) NFKB1NFKB2RELAKDM1ABTK
SCHEMBL13628664 0.86 NFKB1 (0.51) NFKB1NFKB2RELAKDM1ABTK
SCHEMBL5545237 0.85 NFKB1 (0.50) NFKB1NFKB2RELAKDM1ABTK
SCHEMBL14511588 0.85 NFKB1 (0.50) NFKB1NFKB2RELAKDM1ABTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7071175-B1 Pyridine mercapto carboxylic acids as carboxypeptidase U inhibitors ASTRAZENECA AB (SE) 2006-07-04 US disclosed
EP-1180098-A1 NEW COMPOUNDS AstraZeneca AB (SE) 2002-02-20 EP disclosed
WO-2000066557-A1 NEW COMPOUNDS ASTRAZENECA AB (SE) 2000-11-09 WO disclosed