SCHEMBL6059031

SCHEMBL6059031

C=Cc1cc(C(=O)OCC)cnc1N(C(=O)OC(C)(C)C)C(=O)OC(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
SYK P43405 1/20 0.37
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
MAPT P10636 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
MEN1 O00255 1/20 0.36
MAPK1 P28482 1/20 0.36
KMT2A Q03164 1/20 0.36
CA12 O43570 2/20 0.34
CA1 P00915 2/20 0.34
CA2 P00918 2/20 0.34
CA7 P43166 2/20 0.34
CA9 Q16790 2/20 0.34
CA14 Q9ULX7 2/20 0.34
MAOB P27338 3/20 0.34
PDPK1 O15530 1/20 0.34
ALDH1A1 P00352 2/20 0.33
NFKB1 P19838 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6059549 0.82 SYK (0.44) CYP2C9CYP2C19SYKMAPK1KMT2A
SCHEMBL6059213 0.82 CYP2C19 (0.41) CYP2C9CYP2C19SYKNPC1RAB9A
SCHEMBL23501684 0.76 CYP2C9 (0.49) CYP2C9CYP2C19NPC1RAB9AMEN1
SCHEMBL1092469 0.75 CYP2C9 (0.51) CYP2C9CYP2C19NPC1RAB9ASMN1; SMN2
SCHEMBL16649767 0.74 CYP2C19 (0.40) CYP2C9CYP2C19SYKNPC1RAB9A
SCHEMBL465766 0.74 SYK (0.47) CYP2C9CYP2C19SYKNPC1RAB9A
SCHEMBL16421764 0.74 CYP2C9 (0.47) CYP2C9CYP2C19NPC1RAB9AMAPT
SCHEMBL31405437 0.74 CYP2C9 (0.47) CYP2C9CYP2C19NPC1RAB9AMEN1
SCHEMBL4039418 0.73 CYP2C19 (0.57) CYP2C9CYP2C19SYKNPC1RAB9A
SCHEMBL19266065 0.72 CYP2C9 (0.44) CYP2C9CYP2C19NPC1RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7071175-B1 Pyridine mercapto carboxylic acids as carboxypeptidase U inhibitors ASTRAZENECA AB (SE) 2006-07-04 US disclosed
EP-1180098-A1 NEW COMPOUNDS AstraZeneca AB (SE) 2002-02-20 EP disclosed
WO-2000066557-A1 NEW COMPOUNDS ASTRAZENECA AB (SE) 2000-11-09 WO disclosed