SCHEMBL6059293

SCHEMBL6059293

C=C(Cc1ccc(NC(=O)OC(C)(C)C)nc1C)C(=O)OCC

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LCK P06239 4/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34
SCN9A Q15858 1/20 0.33
CYP17A1 P05093 2/20 0.33
ALDH1A1 P00352 1/20 0.33
PTGER1 P34995 1/20 0.32
GSK3B P49841 1/20 0.32
DYRK1A Q13627 1/20 0.32
ALOX15 P16050 1/20 0.32
KMT2A Q03164 1/20 0.32
MKNK2 Q9HBH9 1/20 0.32
P2RX7 Q99572 1/20 0.32
MAPKAPK2 P49137 1/20 0.32
PI4KB Q9UBF8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Diethylamine SCHEMBL7375183 0.96 LCK (0.32) LCKPTGDR2SCN9ACYP17A1ALDH1A1
SCHEMBL3820976 0.80 NAMPT (0.43) PTGDR2SCN9ACYP17A1ALDH1A1GSK3B
SCHEMBL6059133 0.79 ALDH1A1 (0.36) LCKSCN9ACYP17A1ALDH1A1PTGER1
SCHEMBL6059352 0.79 LCK (0.40) LCKPTGDR2SCN9ACYP17A1PTGER1
SCHEMBL3888187 0.78 LCK (0.39) LCKPTGDR2SCN9ACYP17A1PTGER1
SCHEMBL6059214 0.78 LCK (0.39) LCKPTGDR2SCN9ACYP17A1PTGER1
SCHEMBL6059061 0.77 PPARG (0.37) LCKPTGDR2SCN9ACYP17A1ALDH1A1
SCHEMBL6058901 0.76 IGF1R (0.41) CYP17A1ALDH1A1MKNK2
Diethylamine SCHEMBL7380494 0.76 NAMPT (0.41) PTGDR2SCN9ACYP17A1ALDH1A1GSK3B
SCHEMBL28085713 0.76 ALDH1A1 (0.48) ALDH1A1ALOX15KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7071175-B1 Pyridine mercapto carboxylic acids as carboxypeptidase U inhibitors ASTRAZENECA AB (SE) 2006-07-04 US disclosed
EP-1180098-A1 NEW COMPOUNDS AstraZeneca AB (SE) 2002-02-20 EP disclosed
WO-2000066557-A1 NEW COMPOUNDS ASTRAZENECA AB (SE) 2000-11-09 WO disclosed