SCHEMBL6059375

SCHEMBL6059375

CC/C=C(\Cc1ccc(NC(=O)OC(C)(C)C)nc1)C(=O)OCC

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.41
HDAC1 Q13547 1/20 0.41
NPSR1 Q6W5P4 1/20 0.38
MKNK2 Q9HBH9 1/20 0.38
GRIN2B Q13224 1/20 0.37
KDM4E B2RXH2 1/20 0.36
HPGD P15428 1/20 0.36
MAPT P10636 2/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP17A1 P05093 1/20 0.35
POLB P06746 1/20 0.35
GAA P10253 1/20 0.35
GSK3B P49841 1/20 0.35
DYRK1A Q13627 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.35
RAB9A P51151 2/20 0.34
WNT3A P56704 2/20 0.34
SCN9A Q15858 1/20 0.34
PPARG P37231 2/20 0.33
PPARA Q07869 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6058862 1.00 NAMPT (0.41) NAMPTHDAC1NPSR1MKNK2GRIN2B
SCHEMBL6059332 0.92 NAMPT (0.40) NAMPTHDAC1NPSR1MKNK2GRIN2B
SCHEMBL6059113 0.91 NAMPT (0.42) NAMPTHDAC1NPSR1MKNK2GRIN2B
SCHEMBL6059117 0.91 NAMPT (0.42) NAMPTHDAC1NPSR1MKNK2GRIN2B
SCHEMBL3820976 0.84 NAMPT (0.43) NAMPTHDAC1NPSR1MKNK2GRIN2B
SCHEMBL2871142 0.83 NAMPT (0.46) NAMPTHDAC1MKNK2GRIN2BKDM4E
SCHEMBL6059329 0.81 NAMPT (0.41) NAMPTHDAC1NPSR1MKNK2GRIN2B
Diethylamine SCHEMBL7380494 0.80 NAMPT (0.41) NAMPTHDAC1NPSR1MKNK2GRIN2B
SCHEMBL949620 0.78 NAMPT (0.48) NAMPTHDAC1GRIN2BMAPTCYP17A1
SCHEMBL15354526 0.78 NAMPT (0.50) NAMPTHDAC1MKNK2GRIN2BCYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7071175-B1 Pyridine mercapto carboxylic acids as carboxypeptidase U inhibitors ASTRAZENECA AB (SE) 2006-07-04 US disclosed
EP-1180098-A1 NEW COMPOUNDS AstraZeneca AB (SE) 2002-02-20 EP disclosed
WO-2000066557-A1 NEW COMPOUNDS ASTRAZENECA AB (SE) 2000-11-09 WO disclosed