SCHEMBL6061289

SCHEMBL6061289

Cc1nc2c3c(ccn2c1C)C(O)CC(c1cccc(Cl)c1Cl)N3

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.33
CYP2C9 P11712 2/20 0.33
LMNA P02545 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
GBA1 P04062 1/20 0.31
PTPN11 Q06124 2/20 0.30
MEN1 O00255 1/20 0.30
GAA P10253 1/20 0.30
KMT2A Q03164 1/20 0.30
OPRM1 P35372 2/20 0.30
OPRL1 P41146 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1818094 0.92 CYP3A4 (0.36) CYP3A4CYP2C9L3MBTL1GAA
SCHEMBL1814419 0.90 CYP3A4 (0.35) CYP3A4CYP2C9OPRM1OPRL1
SCHEMBL1814676 0.81 CYP3A4 (0.46) CYP3A4CYP2C9
SCHEMBL1816294 0.80 CYP3A4 (0.35) CYP3A4CYP2C9L3MBTL1GBA1GAA
SCHEMBL4885373 0.76 CYP3A4 (0.36) CYP3A4CYP2C9
SCHEMBL4887936 0.76 CYP3A4 (0.34) CYP3A4CYP2C9
SCHEMBL5634862 0.69 CYP3A4 (0.41) CYP3A4CYP2C9KMT2A
SCHEMBL5634281 0.69 CYP3A4 (0.41) CYP3A4CYP2C9LMNAL3MBTL1GAA
SCHEMBL10921468 0.65 ATP4A (0.51) CYP3A4CYP2C9
SCHEMBL7142034 0.65 CYP3A4 (0.38) CYP3A4CYP2C9GBA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1663313-A2 COMPOSITIONS USEFUL FOR TREATING GASTROINTESTINAL MOTILITY DISORDERS Dynogen Pharmaceuticals Inc. (US) 2006-06-07 EP disclosed
WO-2005021040-A2 COMPOSITIONS USEFUL FOR TREATING GASTROINTESTINAL MOTILITY DISORDERS DYNOGEN PHARMACEUTICALS, INC. (US) 2005-03-10 WO disclosed