SCHEMBL6063528

SCHEMBL6063528

COc1ccc(-c2cnc3nc(N)nc(N(C(C)O)C(C)O)c3n2)cc1OC

nearest known ligand 0.68

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 9/20 0.68
PIK3CG P48736 3/20 0.44
SYK P43405 1/20 0.42
GAK O14976 1/20 0.41
STK17B O94768 1/20 0.41
PIK3CA P42336 2/20 0.41
PIK3CB P42338 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
NEK2 P51955 1/20 0.39
MAPK1 P28482 1/20 0.39
MAPK8 P45983 1/20 0.39
MAPK9 P45984 1/20 0.39
MAPK10 P53779 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5523882 0.85 NOS1 (0.74) NOS1PIK3CGGAKSTK17BPIK3CA
SCHEMBL5513759 0.83 NOS1 (0.84) NOS1PIK3CGGAK
Water SCHEMBL6483778 0.82 NOS1 (0.82) NOS1PIK3CGGAK
SCHEMBL5513505 0.81 NOS1 (1.00) NOS1PIK3CGGAK
SCHEMBL6063542 0.81 NOS1 (0.67) NOS1PIK3CGSYKGAKSTK17B
Water SCHEMBL6483075 0.80 NOS1 (0.98) NOS1PIK3CGGAK
SCHEMBL4454683 0.79 NOS1 (0.60) NOS1PIK3CGSYKGAKSTK17B
SCHEMBL4449231 0.79 NOS1 (0.60) NOS1PIK3CGSYKGAKSTK17B
SCHEMBL5508808 0.78 NOS1 (1.00) NOS1PIK3CGMAPK1
SCHEMBL5514530 0.78 NOS1 (0.59) NOS1PIK3CGSYKGAKSTK17B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1658081-A2 IMMUNOSUPPRESSIVE EFFECTS OF PTERIDINE DERIVATIVES 4 AZA Bioscience nv (BE) 2006-05-24 EP claimed
WO-2005021003-A2 IMMUNOSUPPRESSIVE EFFECTS OF PTERIDINE DERIVATIVES 4 AZA BIOSCIENCE NV (BE) 2005-03-10 WO claimed