SCHEMBL6063751

SCHEMBL6063751

CC(C)Oc1nc(N)nc2ncc(-c3ccc(F)c(F)c3)nc12.COc1ccc(-c2cnc3nc(N)nc(OC(C)C)c3n2)cc1

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 9/20 0.53
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43
XDH P47989 1/20 0.43
DYRK1A Q13627 1/20 0.42
POLB P06746 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
PIK3CG P48736 2/20 0.39
KDM4E B2RXH2 1/20 0.38
ALOX5AP P20292 1/20 0.38
FEN1 P39748 1/20 0.38
SGK1 O00141 1/20 0.38
PIK3CA P42336 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4448850 0.93 PIK3CG (0.44) NOS1ALDH1A1PIK3CGALOX5APFEN1
SCHEMBL5510798 0.91 NOS1 (0.63) NOS1ALDH1A1HPGDXDHDYRK1A
SCHEMBL4455139 0.83 PIK3CG (0.42) NOS1PIK3CGALOX5APFEN1PIK3CA
SCHEMBL3757292 0.83 NOS1 (0.49) NOS1PIK3CGALOX5APFEN1PIK3CA
SCHEMBL4451388 0.82 NOS1 (0.54) NOS1ALDH1A1HPGDXDHDYRK1A
SCHEMBL4449231 0.81 NOS1 (0.60) NOS1PIK3CGPIK3CA
SCHEMBL4451834 0.80 NOS1 (0.51) NOS1L3MBTL1PIK3CGKDM4EPIK3CA
SCHEMBL4453670 0.80 NOS1 (0.52) NOS1ALDH1A1PIK3CGKDM4E
SCHEMBL4454718 0.79 PIK3CG (0.45) NOS1HPGDPIK3CGPIK3CA
SCHEMBL3757239 0.79 NOS1 (0.46) NOS1ALDH1A1PIK3CGPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1658081-A2 IMMUNOSUPPRESSIVE EFFECTS OF PTERIDINE DERIVATIVES 4 AZA Bioscience nv (BE) 2006-05-24 EP claimed
WO-2005021003-A2 IMMUNOSUPPRESSIVE EFFECTS OF PTERIDINE DERIVATIVES 4 AZA BIOSCIENCE NV (BE) 2005-03-10 WO claimed