SCHEMBL6064082

SCHEMBL6064082

CCNc1nc(N)nc2ncc(-c3ccc(OC)c(OC)c3)nc12.c1cc2ccc1-2

nearest known ligand 0.63

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 5/20 0.63
STK17B O94768 1/20 0.46
MAPK1 P28482 1/20 0.44
PIK3CA P42336 1/20 0.44
MAPK8 P45983 1/20 0.44
MAPK9 P45984 1/20 0.44
MAPK10 P53779 1/20 0.44
DHFR P00374 3/20 0.44
BRAF P15056 1/20 0.43
HPGD P15428 1/20 0.42
PIK3CG P48736 1/20 0.42
GAK O14976 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5516964 0.90 NOS1 (0.65) NOS1STK17BMAPK1PIK3CAMAPK8
SCHEMBL6063982 0.85 NOS1 (0.69) NOS1DHFRHPGD
SCHEMBL6063923 0.84 NOS1 (0.60) NOS1STK17BMAPK1PIK3CAMAPK8
SCHEMBL6062659 0.84 NOS1 (0.60) NOS1STK17BMAPK1PIK3CAMAPK8
SCHEMBL6062674 0.84 NOS1 (0.60) NOS1STK17BMAPK1PIK3CAMAPK8
SCHEMBL6064072 0.84 NOS1 (0.65) NOS1MAPK1HPGD
SCHEMBL6063556 0.82 NOS1 (0.55) NOS1MAPK1DHFRHPGD
SCHEMBL4454283 0.81 NOS1 (0.67) NOS1MAPK1PIK3CAMAPK8MAPK9
SCHEMBL6815729 0.80 NOS1 (0.60) NOS1STK17BBRAFHPGDGAK
SCHEMBL5513759 0.79 NOS1 (0.84) NOS1PIK3CGGAK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1658081-A2 IMMUNOSUPPRESSIVE EFFECTS OF PTERIDINE DERIVATIVES 4 AZA Bioscience nv (BE) 2006-05-24 EP claimed
WO-2005021003-A2 IMMUNOSUPPRESSIVE EFFECTS OF PTERIDINE DERIVATIVES 4 AZA BIOSCIENCE NV (BE) 2005-03-10 WO claimed