SCHEMBL6065336

SCHEMBL6065336

COc1c(CCN2CCN(c3cccc4nc(C)ccc34)CC2)cccc1N1CCN(C)C1=O

nearest known ligand 0.61

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 18/20 0.61
HTR1D P28221 18/20 0.61
HTR1B P28222 18/20 0.61
SLC6A4 P31645 15/20 0.61
KCNH2 Q12809 15/20 0.61
CYP2C9 P11712 3/20 0.57
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
DRD2 P14416 1/20 0.52
HTR2A P28223 1/20 0.52
HTR2C P28335 1/20 0.52
CYP2C19 P33261 1/20 0.52
HTR7 P34969 1/20 0.52
DRD3 P35462 1/20 0.52
HTR2B P41595 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL2884146 0.99 HTR1A (0.60) HTR1AHTR1DHTR1BSLC6A4KCNH2
SCHEMBL2883396 0.87 HTR1A (0.67) HTR1AHTR1DHTR1BSLC6A4KCNH2
Hydrochloric Acid SCHEMBL2878647 0.86 HTR1A (0.66) HTR1AHTR1DHTR1BSLC6A4KCNH2
Hydrochloric Acid SCHEMBL2897763 0.85 HTR1A (0.67) HTR1AHTR1DHTR1BSLC6A4KCNH2
SCHEMBL2881169 0.85 CYP2C9 (0.64) HTR1AHTR1DHTR1BSLC6A4KCNH2
SCHEMBL2883222 0.81 HTR1A (0.59) HTR1AHTR1DHTR1BSLC6A4KCNH2
SCHEMBL2882984 0.80 HTR1D (0.76) HTR1AHTR1DHTR1BSLC6A4KCNH2
Hydrochloric Acid SCHEMBL2883364 0.79 HTR1A (0.63) HTR1AHTR1DHTR1BSLC6A4KCNH2
Hydrochloric Acid SCHEMBL2882627 0.79 HTR1A (0.63) HTR1AHTR1DHTR1BSLC6A4KCNH2
SCHEMBL6065950 0.78 CYP2C9 (0.73) HTR1AHTR1DHTR1BSLC6A4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1646613-A1 QUINOLINE AND QUINAZOLINE DERIVATIVES HAVING AFFINITY FOR 5HT1-TYPE RECEPTORS GLAXO GROUP LIMITED (GB) 2006-04-19 EP disclosed
WO-2005014552-A1 QUINOLINE AND QUINAZOLINE DERIVATIVES HAVING AFFINITY FOR 5HT1-TYPE RECEPTORS GLAXO GROUP LIMITED (GB) 2005-02-17 WO disclosed