SCHEMBL6065404

SCHEMBL6065404

O=C(Cc1cccc2cnccc12)NCCC(F)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ROS1 P08922 1/20 0.51
RPS6KB1 P23443 1/20 0.51
TRPV1 Q8NER1 15/20 0.50
GLS O94925 1/20 0.43
DGAT2 Q96PD7 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6066295 0.90 ROS1 (0.53) ROS1RPS6KB1TRPV1GLSDGAT2
SCHEMBL4026467 0.82 ROS1 (0.73) ROS1RPS6KB1TRPV1DGAT2
SCHEMBL4020324 0.79 EPHX2 (0.60) ROS1RPS6KB1TRPV1GLS
SCHEMBL4030337 0.78 TRPV1 (0.69) ROS1RPS6KB1TRPV1GLSDGAT2
SCHEMBL4021187 0.77 TRPV1 (0.57) ROS1RPS6KB1TRPV1GLSDGAT2
SCHEMBL4021335 0.76 ROS1 (0.55) ROS1RPS6KB1TRPV1DGAT2
SCHEMBL4022317 0.72 ROS1 (0.61) ROS1RPS6KB1TRPV1GLS
SCHEMBL4025364 0.72 TRPV1 (0.64) ROS1RPS6KB1TRPV1GLS
SCHEMBL6583327 0.72 ROS1 (0.55) ROS1RPS6KB1TRPV1GLS
SCHEMBL4022175 0.72 ROS1 (0.73) ROS1RPS6KB1TRPV1GLS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1660455-A1 FUSED AZABICYCLIC COMPOUNDS THAT INHIBIT VANILLOID RECEPTOR SUBTYPE 1 (VR1) RECEPTOR ABBOTT LABORATORIES (US) 2006-05-31 EP disclosed
WO-2005016890-A1 FUSED AZABICYCLIC COMPOUNDS THAT INHIBIT VANILLOID RECEPTOR SUBTYPE 1 (VR1) RECEPTOR ABBOTT LABORATORIES (US) 2005-02-24 WO disclosed