SCHEMBL6583327

SCHEMBL6583327

O=C(Cc1cccc2cnccc12)NCCc1ccc(C(F)(F)F)c(F)c1

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ROS1 P08922 1/20 0.55
RPS6KB1 P23443 1/20 0.55
TRPV1 Q8NER1 14/20 0.51
PTPN1 P18031 1/20 0.45
GLS O94925 1/20 0.44
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPT P10636 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
P2RX7 Q99572 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6587146 0.94 ROS1 (0.53) ROS1RPS6KB1TRPV1GLSKDM4E
SCHEMBL4030518 0.91 ROS1 (0.64) ROS1RPS6KB1TRPV1GLSKDM4E
SCHEMBL4030337 0.85 TRPV1 (0.69) ROS1RPS6KB1TRPV1PTPN1GLS
SCHEMBL6584430 0.83 TRPV1 (0.74) TRPV1
SCHEMBL4019570 0.80 ROS1 (0.69) ROS1RPS6KB1TRPV1GLSKDM4E
SCHEMBL4025364 0.80 TRPV1 (0.64) ROS1RPS6KB1TRPV1PTPN1GLS
SCHEMBL5391279 0.79 ROS1 (0.81) ROS1RPS6KB1TRPV1PTPN1GLS
SCHEMBL4021307 0.79 ROS1 (0.63) ROS1RPS6KB1TRPV1PTPN1GLS
SCHEMBL4023632 0.79 ROS1 (0.57) ROS1RPS6KB1TRPV1GLSKDM4E
SCHEMBL4023210 0.78 TRPV1 (0.69) ROS1RPS6KB1TRPV1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1478363-A1 FUSED AZABICYCLIC COMPOUNDS THAT INHIBIT VANILLOID RECEPTOR SUBTYPE 1 (VR1) RECEPTOR Abbott Laboratories (US) 2004-11-24 EP claimed
WO-2003070247-A1 FUSED AZABICYCLIC COMPOUNDS THAT INHIBIT VANILLOID RECEPTOR SUBTYPE 1 (VR1) RECEPTOR ABBOTT LABORATORIES (US) 2003-08-28 WO claimed