SCHEMBL6068348

SCHEMBL6068348

CCOC(=O)CNC(=O)N1CCN(c2cc(N(C)Cc3cccnc3)nc(Nc3nc(C)c(C(=O)OCC)s3)n2)CC1

nearest known ligand 0.58

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 6/20 0.58
TP53 P04637 1/20 0.42
ALDH1A1 P00352 4/20 0.40
MAPT P10636 4/20 0.40
KDM4E B2RXH2 3/20 0.40
LMNA P02545 2/20 0.39
NPC1 O15118 1/20 0.38
HPGD P15428 1/20 0.38
RAB9A P51151 1/20 0.38
DHODH Q02127 3/20 0.38
CSNK1D P48730 1/20 0.38
CYP17A1 P05093 1/20 0.37
CYP21A2 P08686 1/20 0.37
CYP11B1 P15538 1/20 0.37
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29408543 1.00 PDE5A (0.58) PDE5ATP53ALDH1A1MAPTKDM4E
SCHEMBL2696718 0.95 PDE5A (0.52) PDE5ATP53ALDH1A1MAPTKDM4E
SCHEMBL28565216 0.89 PDE5A (0.73) PDE5ATP53ALDH1A1MAPTKDM4E
SCHEMBL29408541 0.89 PDE5A (0.73) PDE5ATP53ALDH1A1MAPTKDM4E
SCHEMBL6068425 0.88 PDE5A (0.57) PDE5ATP53ALDH1A1MAPTKDM4E
SCHEMBL29408493 0.88 PDE5A (0.57) PDE5ATP53ALDH1A1MAPTKDM4E
SCHEMBL2680815 0.87 PDE5A (0.73) PDE5ATP53ALDH1A1MAPTKDM4E
SCHEMBL29408511 0.86 PDE5A (0.69) PDE5ATP53ALDH1A1MAPTKDM4E
SCHEMBL6068350 0.86 PDE5A (0.69) PDE5ATP53ALDH1A1MAPTKDM4E
SCHEMBL6068408 0.86 PDE5A (0.60) PDE5ATP53ALDH1A1MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7087614-B2 Pyrimidine inhibitors of phosphodiesterase (PDE) 7 BRISTOL-MYERS SQUIBB CO. (US) 2006-08-08 US disclosed