SCHEMBL6068424

SCHEMBL6068424

COc1cc(CNc2cc(N3CCC(O)C(O)C3C)nc(Nc3nc(C)c(C(=O)O)s3)n2)cc(OC)c1OC

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 7/20 0.49
PDE2A O00408 1/20 0.36
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
ACHE P22303 1/20 0.36
BACE1 P56817 1/20 0.36
ALDH1A1 P00352 4/20 0.35
MAPT P10636 2/20 0.35
TSHR P16473 1/20 0.35
KDM4E B2RXH2 1/20 0.35
LMNA P02545 2/20 0.33
HIF1A Q16665 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
ALK Q9UM73 2/20 0.33
IGF1R P08069 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
CCNT1 O60563 1/20 0.32
CCNE1 P24864 1/20 0.32
CDK2 P24941 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL289823 0.86 PDE5A (0.58) PDE5APDE2APDE3BPDE3AACHE
SCHEMBL290933 0.85 PDE5A (0.54) PDE5APDE2APDE3BPDE3AACHE
SCHEMBL290275 0.84 PDE5A (0.57) PDE5APDE2APDE3BPDE3AACHE
SCHEMBL6068433 0.83 PDE5A (0.58) PDE5AALDH1A1MAPTTSHRKDM4E
SCHEMBL291065 0.83 PDE5A (0.58) PDE5APDE2APDE3BPDE3AACHE
SCHEMBL26647635 0.83 PDE5A (0.62) PDE5APDE2APDE3BPDE3A
SCHEMBL291323 0.82 PDE5A (0.56) PDE5APDE2APDE3BPDE3AACHE
SCHEMBL291180 0.81 PDE5A (0.54) PDE5AALKIGF1R
SCHEMBL291049 0.81 PDE5A (0.54) PDE5AALKIGF1R
SCHEMBL291168 0.79 PDE5A (0.52) PDE5APDE2APDE3BPDE3AACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7087614-B2 Pyrimidine inhibitors of phosphodiesterase (PDE) 7 BRISTOL-MYERS SQUIBB CO. (US) 2006-08-08 US disclosed