SCHEMBL6072290

SCHEMBL6072290

CCOC(=O)CNC(=O)c1ccc(C2=NC(C)(C)Cc3cc(OCC)c4c(c32)CC(C)(C)O4)cc1NCc1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPID Q08752 2/20 0.36
POLB P06746 1/20 0.35
HTT P42858 1/20 0.33
KMT2A Q03164 3/20 0.33
MEN1 O00255 2/20 0.33
RAB9A P51151 2/20 0.33
NPC1 O15118 1/20 0.33
EZH2 Q15910 1/20 0.32
TSHR P16473 1/20 0.32
HBB P68871 1/20 0.32
CDC7 O00311 1/20 0.32
ROCK2 O75116 1/20 0.32
MAP4K4 O95819 1/20 0.32
GSK3B P49841 1/20 0.32
CLK4 Q9HAZ1 1/20 0.32
MKNK2 Q9HBH9 1/20 0.32
HPGD P15428 2/20 0.32
ALDH1A1 P00352 4/20 0.32
L3MBTL1 Q9Y468 2/20 0.32
BRCA1 P38398 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6072007 0.94 POLB (0.36) POLBKMT2AMEN1RAB9ANPC1
Hydrochloric Acid SCHEMBL6072454 0.92 CDC7 (0.35) POLBKMT2AMEN1RAB9ANPC1
SCHEMBL6071853 0.91 NPSR1 (0.38) POLBHTTKMT2AMEN1RAB9A
SCHEMBL6072319 0.91 HTT (0.36) POLBHTTKMT2AMEN1ALDH1A1
SCHEMBL6072191 0.89 ACLY (0.38) POLBHTTKMT2AMEN1RAB9A
SCHEMBL6072328 0.89 POLB (0.32) POLBKMT2ARAB9ANPC1TSHR
Hydrochloric Acid SCHEMBL6072323 0.89 POLB (0.32) POLBRAB9ANPC1CDC7ROCK2
SCHEMBL6072162 0.89 MKNK2 (0.42) POLBRAB9ANPC1CDC7ROCK2
Hydrochloric Acid SCHEMBL6072452 0.88 CXCR2 (0.34) POLBKMT2AMEN1RAB9ANPC1
SCHEMBL6071890 0.88 POLB (0.36) POLBKMT2AMEN1RAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060106048-A1 Furoisoquinoline derivative and use thereof PASCALI, PETROS P. (CY) 2006-05-18 US disclosed
EP-1541576-A1 FUROISOQUINOLINE DERIVATIVE AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2005-06-15 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060106048-A1 Furoisoquinoline derivative and use thereof PDE3B, PDE2A, PDE3A PPID 4187/4885POLB 1887/4885HTT 4539/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.