SCHEMBL6072947

SCHEMBL6072947

O=C(NCC1C2CN(Cc3ccccc3)CC12)N1CCc2ccccc2C1c1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HHAT Q5VTY9 3/20 0.47
CYP2D6 P10635 1/20 0.46
GRIN1 Q05586 1/20 0.46
GRIN2B Q13224 1/20 0.46
SIGMAR1 Q99720 1/20 0.46
TRPM8 Q7Z2W7 5/20 0.45
HDAC8 Q9BY41 1/20 0.44
CHRM3 P20309 2/20 0.44
CACNA1F O60840 1/20 0.44
CHRM2 P08172 1/20 0.44
CHRM4 P08173 1/20 0.44
CHRM5 P08912 1/20 0.44
CHRM1 P11229 1/20 0.44
KCNE1 P15382 1/20 0.44
KCNQ1 P51787 1/20 0.44
CACNA1D Q01668 1/20 0.44
KCNH2 Q12809 1/20 0.44
CACNA1S Q13698 1/20 0.44
CACNA1C Q13936 1/20 0.44
SCN5A Q14524 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6072959 0.87 CHRM3 (0.50) HHATCYP2D6GRIN1GRIN2BSIGMAR1
SCHEMBL6073422 0.84 HHAT (0.51) HHATCYP2D6TRPM8HDAC8
SCHEMBL6072987 0.83 CHRM3 (0.52) HHATCYP2D6GRIN1GRIN2BSIGMAR1
SCHEMBL17117236 0.79 HHAT (0.54) HHATCYP2D6TRPM8HDAC8
SCHEMBL17117340 0.77 EPHX2 (0.58) HHATCYP2D6TRPM8HDAC8
SCHEMBL6072890 0.74 CHRM3 (0.61) HHATCYP2D6GRIN1GRIN2BSIGMAR1
SCHEMBL1014404 0.74 S1PR5 (0.50) GRIN2BSIGMAR1
SCHEMBL4924735 0.73 TSHR (0.48) GRIN1GRIN2BSIGMAR1
SCHEMBL6073004 0.72 CHRM3 (0.52) HHATCYP2D6TRPM8HDAC8CHRM3
SCHEMBL22776336 0.72 CHRM3 (0.57) HHATTRPM8CHRM3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006035280-A1 3,4-DIHYDROISOQUINOLINE COMPOUNDS AS MUSCRINIC RECEPTOR ANTAGONISTS FOR THE TREATMENT OF RESPIRATORY, URINARY AND GASTROINTESTINAL DISEASES RANBAXY LABORATORIES LIMITED (IN) 2006-04-06 WO claimed