SCHEMBL6073422

SCHEMBL6073422

O=C(NCC1C2CNCC21)N1CCc2ccccc2C1c1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HHAT Q5VTY9 3/20 0.51
CYP2D6 P10635 1/20 0.50
HDAC8 Q9BY41 2/20 0.48
TRPM8 Q7Z2W7 9/20 0.47
HDAC3 O15379 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC2 Q92769 1/20 0.47
NCOR2 Q9Y618 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6073004 0.85 CHRM3 (0.52) HHATCYP2D6HDAC8TRPM8
SCHEMBL6072947 0.84 HHAT (0.47) HHATCYP2D6HDAC8TRPM8
SCHEMBL6072963 0.82 CHRM3 (0.53) HHATCYP2D6HDAC8HDAC3HDAC1
SCHEMBL22784521 0.81 CHRM3 (0.60) TRPM8
Acetic Acid SCHEMBL22776782 0.79 CHRM3 (0.56) HHATCYP2D6TRPM8
Acetic Acid SCHEMBL29560775 0.79 CHRM3 (0.56) HHATCYP2D6TRPM8
SCHEMBL17117236 0.78 HHAT (0.54) HHATCYP2D6HDAC8TRPM8HDAC3
SCHEMBL22776219 0.77 TRPM8 (0.55) TRPM8
SCHEMBL22776218 0.77 TRPM8 (0.55) TRPM8
SCHEMBL22784205 0.77 TRPM8 (0.55) TRPM8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006035280-A1 3,4-DIHYDROISOQUINOLINE COMPOUNDS AS MUSCRINIC RECEPTOR ANTAGONISTS FOR THE TREATMENT OF RESPIRATORY, URINARY AND GASTROINTESTINAL DISEASES RANBAXY LABORATORIES LIMITED (IN) 2006-04-06 WO claimed
WO-2006035280-A1 3,4-DIHYDROISOQUINOLINE COMPOUNDS AS MUSCRINIC RECEPTOR ANTAGONISTS FOR THE TREATMENT OF RESPIRATORY, URINARY AND GASTROINTESTINAL DISEASES RANBAXY LABORATORIES LIMITED (IN) 2006-04-06 WO disclosed