SCHEMBL6073344

SCHEMBL6073344

CSc1ncc2cc(Br)c(N)nc2n1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 5/20 0.40
HASPIN Q8TF76 1/20 0.38
KMT2A Q03164 3/20 0.36
HTT P42858 2/20 0.36
AKT1 P31749 7/20 0.33
AKT2 P31751 7/20 0.33
POLB P06746 1/20 0.32
RAB9A P51151 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
MEN1 O00255 2/20 0.32
SRC P12931 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29742257 1.00 FGFR1 (0.40) FGFR1HASPINKMT2AHTTAKT1
SCHEMBL6073526 0.81 FGFR1 (0.42) FGFR1HASPINKMT2AHTTAKT1
SCHEMBL16683500 0.81 MEN1 (0.35) HASPINKMT2AHTTAKT1AKT2
SCHEMBL6073377 0.80 MEN1 (0.38) HASPINKMT2AHTTAKT1AKT2
SCHEMBL29537852 0.80 MEN1 (0.38) HASPINKMT2AHTTAKT1AKT2
SCHEMBL25225563 0.80 MEN1 (0.35) HASPINKMT2AAKT1AKT2MEN1
SCHEMBL3293161 0.80 MEN1 (0.41) FGFR1HASPINKMT2AAKT1AKT2
SCHEMBL6073568 0.80 HASPIN (0.38) FGFR1HASPINKMT2AAKT1AKT2
SCHEMBL29537604 0.80 MEN1 (0.35) HASPINKMT2AAKT1AKT2MEN1
SCHEMBL31344333 0.80 HASPIN (0.36) FGFR1HASPINKMT2AAKT1AKT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7053070-B2 Pyrido[2,3-d]pyrimidine-2,7-diamine kinase inhibitors WARNER-LAMBERT COMPANY (US) 2006-05-30 US disclosed
US-20030073668-A1 Pyrido[2,3-d]pyrimidine-2,7-diamine kinase inhibitors BOOTH RICHARD JOHN (US) 2003-04-17 US disclosed
EP-1254137-A1 PYRIDO 2,3-d]PYRIMIDINE-2,7-DIAMINE KINASE INHIBITORS WARNER-LAMBERT COMPANY (US) 2002-11-06 EP disclosed
WO-2001055147-A1 PYRIDO[2,3-d]PYRIMIDINE-2,7-DIAMINE KINASE INHIBITORS WARNER-LAMBERT COMPANY (US) 2001-08-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030073668-A1 Pyrido[2,3-d]pyrimidine-2,7-diamine kinase inhibitors CDK9, CDK19, CDK3 FGFR1 280/4885HASPIN 3207/4885KMT2A 2672/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.