SCHEMBL6075770

SCHEMBL6075770

Cc1ccc(-c2nc3c(c(NC4CCC(C)CC4)n2)CCCC3)cc1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 1/20 0.45
MAPT P10636 2/20 0.42
TP53 P04637 1/20 0.42
GBA1 P04062 1/20 0.40
ALDH1A1 P00352 2/20 0.39
HPGD P15428 1/20 0.39
HTT P42858 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
ACP1 P24666 1/20 0.39
IGF1R P08069 1/20 0.38
PDE4B Q07343 2/20 0.38
PTGS2 P35354 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38
CLK4 Q9HAZ1 1/20 0.38
TLR9 Q9NR96 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6075144 0.95 ACP1 (0.42) ADORA1MAPTALDH1A1HPGDHTT
SCHEMBL6075371 0.91 IGF1R (0.42) ADORA1MAPTALDH1A1HPGDHTT
SCHEMBL6076160 0.91 ACP1 (0.45) ADORA1MAPTALDH1A1HPGDHTT
SCHEMBL6076928 0.90 PDE5A (0.46) ADORA1MAPTALDH1A1HPGDHTT
SCHEMBL6075878 0.89 ADORA1 (0.47) ADORA1MAPTTP53ALDH1A1HPGD
SCHEMBL6075874 0.89 ADORA1 (0.47) ADORA1MAPTTP53ALDH1A1HPGD
SCHEMBL5732654 0.89 ACP1 (0.45) ADORA1MAPTALDH1A1HPGDHTT
SCHEMBL5734979 0.88 PDE5A (0.46) ADORA1GBA1ACP1IGF1RPDE4B
SCHEMBL5732459 0.87 ADORA1 (0.47) ADORA1MAPTALDH1A1HPGDHTT
SCHEMBL5732457 0.87 ADORA1 (0.47) ADORA1MAPTALDH1A1HPGDHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7045526-B2 Substituted 4-amino-2-aryl-tetrahydroquinazolines, their preparation, their use and pharmaceutical preparations comprising them SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2006-05-16 US claimed