SCHEMBL6075878

SCHEMBL6075878

Cc1ccc(-c2nc3c(c(N[C@H]4CC[C@H](O)CC4)n2)CCCC3)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 4/20 0.47
ADORA2A P29274 3/20 0.47
ADORA3 P0DMS8 2/20 0.45
ADORA2B P29275 1/20 0.45
SGK1 O00141 1/20 0.40
PDE4B Q07343 2/20 0.39
ALDH1A1 P00352 2/20 0.38
HPGD P15428 2/20 0.38
KDM4E B2RXH2 1/20 0.38
MAPT P10636 1/20 0.38
HTT P42858 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
ACP1 P24666 2/20 0.38
IGF1R P08069 1/20 0.38
FLT3 P36888 1/20 0.37
TYRO3 Q06418 1/20 0.37
MERTK Q12866 1/20 0.37
GAS6 Q14393 1/20 0.37
MAPK14 Q16539 1/20 0.37
PTGS2 P35354 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6075874 1.00 ADORA1 (0.47) ADORA1ADORA2AADORA3ADORA2BSGK1
SCHEMBL5732459 0.98 ADORA1 (0.47) ADORA1ADORA2AADORA3ADORA2BSGK1
SCHEMBL5732457 0.98 ADORA1 (0.47) ADORA1ADORA2AADORA3ADORA2BSGK1
SCHEMBL6075144 0.94 ACP1 (0.42) ADORA1ADORA2AADORA3PDE4BALDH1A1
SCHEMBL6075371 0.90 IGF1R (0.42) ADORA1ADORA2AADORA3PDE4BALDH1A1
SCHEMBL6076160 0.90 ACP1 (0.45) ADORA1ADORA2AADORA3PDE4BALDH1A1
SCHEMBL6075770 0.89 ADORA1 (0.45) ADORA1PDE4BALDH1A1HPGDMAPT
SCHEMBL6076928 0.89 PDE5A (0.46) ADORA1ADORA2AADORA3PDE4BALDH1A1
SCHEMBL6076015 0.88 ADORA2A (0.45) ADORA1ADORA2AADORA3ADORA2BSGK1
SCHEMBL6076012 0.88 ADORA2A (0.45) ADORA1ADORA2AADORA3ADORA2BSGK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7045526-B2 Substituted 4-amino-2-aryl-tetrahydroquinazolines, their preparation, their use and pharmaceutical preparations comprising them SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2006-05-16 US claimed