SCHEMBL6079296

SCHEMBL6079296

CC(C)(C)OC(=O)NCCC(Oc1nc(C(F)(F)F)ccc1C#N)C(F)(F)F

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 2/20 0.46
NOS2 P35228 2/20 0.46
AAK1 Q2M2I8 5/20 0.37
TRPA1 O75762 1/20 0.36
BCHE P06276 1/20 0.35
CA12 O43570 5/20 0.35
CA1 P00915 5/20 0.35
CA2 P00918 5/20 0.35
CA9 Q16790 5/20 0.35
AR P10275 1/20 0.35
GPR119 Q8TDV5 1/20 0.34
STING1 Q86WV6 1/20 0.34
MEN1 O00255 1/20 0.34
GAA P10253 1/20 0.34
KMT2A Q03164 1/20 0.34
TRPV1 Q8NER1 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6078734 0.94 SLC6A4 (0.44) SLC6A4NOS2AAK1TRPA1CA12
SCHEMBL6082710 0.82 SLC6A4 (0.46) SLC6A4NOS2AAK1TRPA1AR
SCHEMBL6079471 0.82 SLC6A4 (0.50) SLC6A4NOS2GPR119MEN1KMT2A
SCHEMBL6079478 0.82 SLC6A4 (0.50) SLC6A4NOS2GPR119MEN1KMT2A
SCHEMBL6078732 0.82 SLC6A4 (0.45) SLC6A4NOS2AAK1ARGPR119
SCHEMBL6078728 0.82 SLC6A4 (0.45) SLC6A4NOS2AAK1ARGPR119
Hydrochloric Acid SCHEMBL6079158 0.81 SLC6A4 (0.49) SLC6A4NOS2GPR119MEN1KMT2A
Hydrochloric Acid SCHEMBL6079152 0.81 SLC6A4 (0.49) SLC6A4NOS2GPR119MEN1KMT2A
SCHEMBL6078288 0.76 NOS2 (0.65) SLC6A4NOS2AAK1ARGPR119
Hydrochloric Acid SCHEMBL6077883 0.75 NOS2 (0.64) SLC6A4NOS2AAK1GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7119109-B2 Heteroarylheteroalkylamine derivatives and their use as inhibitors of nitric oxide synthase ASTRAZENECA AB (SE) 2006-10-10 US disclosed