SCHEMBL6081908

SCHEMBL6081908

O=c1n(-c2ccc(OCCNCC3(O)CCCCC3)cc2)ccn1-c1ccc(OC2CCCC2)cc1

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.36
TSHR P16473 1/20 0.36
ADRB1 P08588 2/20 0.35
ADRB3 P13945 2/20 0.35
HRH3 Q9Y5N1 2/20 0.35
RYR2 Q92736 1/20 0.34
HPGD P15428 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
NAAA Q02083 1/20 0.34
HTR1A P08908 1/20 0.33
ADRA1D P25100 1/20 0.33
ADRA1B P35368 1/20 0.33
NPC1 O15118 1/20 0.33
PKM P14618 1/20 0.33
EPHX2 P34913 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6082053 0.84 BTK (0.42) HRH3HTR1AADRA1DADRA1B
SCHEMBL6081904 0.81 HRH3 (0.42) ALDH1A1TSHRHRH3MEN1KMT2A
SCHEMBL1727601 0.81 KDM4E (0.52) ALDH1A1HRH3HPGDMEN1KMT2A
SCHEMBL6081179 0.81 HRH3 (0.41) ALDH1A1HRH3MEN1KMT2ANPC1
SCHEMBL6081508 0.80 KDM4E (0.50) ALDH1A1TSHRHRH3HPGDMEN1
SCHEMBL1728644 0.80 HRH3 (0.42) ALDH1A1TSHRHRH3MEN1KMT2A
SCHEMBL1727849 0.78 KDM4E (0.43) ALDH1A1HRH3
SCHEMBL1728856 0.76 HRH3 (0.42) HRH3
SCHEMBL1729124 0.75 LSS (0.47) HRH3
SCHEMBL1729760 0.75 LSS (0.47) HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7141561-B2 Substituted diaryl heterocycles, process for their preparation and their use as medicaments SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2006-11-28 US disclosed