SCHEMBL6081179

SCHEMBL6081179

COCCCNCCOc1ccc(-n2ccn(-c3ccc(OC4CCCC4)cc3)c2=O)cc1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 5/20 0.41
ACACB O00763 2/20 0.41
KDM4E B2RXH2 6/20 0.41
DRD2 P14416 2/20 0.40
DRD4 P21917 2/20 0.40
DRD3 P35462 2/20 0.40
LMNA P02545 2/20 0.39
ALDH1A1 P00352 2/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
NPC1 O15118 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6081904 0.97 HRH3 (0.42) HRH3ACACBKDM4EDRD2DRD4
SCHEMBL1728644 0.86 HRH3 (0.42) HRH3ACACBKDM4EALDH1A1MEN1
SCHEMBL1727849 0.84 KDM4E (0.43) HRH3ACACBKDM4EALDH1A1CYP1A2
SCHEMBL6081508 0.84 KDM4E (0.50) HRH3KDM4EALDH1A1MEN1KMT2A
SCHEMBL1727601 0.83 KDM4E (0.52) HRH3KDM4EALDH1A1MEN1KMT2A
SCHEMBL6081167 0.83 MCHR1 (0.42) HRH3ACACBKMT2A
SCHEMBL1729087 0.81 MAPK14 (0.51) HRH3KDM4EALDH1A1SMN1; SMN2CYP1A2
SCHEMBL6081908 0.81 ALDH1A1 (0.36) HRH3ALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL1728856 0.80 HRH3 (0.42) HRH3
SCHEMBL1728688 0.80 LSS (0.48) HRH3CYP1A2CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7141561-B2 Substituted diaryl heterocycles, process for their preparation and their use as medicaments SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2006-11-28 US disclosed