SCHEMBL6089729

SCHEMBL6089729

O=C1NN=C(c2ccco2)C1=Cc1cc2c([nH]1)CCCC2=O

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDR P35968 12/20 0.43
PDGFRB P09619 8/20 0.39
FGFR1 P11362 6/20 0.39
SRC P12931 4/20 0.39
PKN1 Q16512 1/20 0.36
PKN2 Q16513 1/20 0.36
BRD4 O60885 1/20 0.35
RET P07949 2/20 0.34
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
HSD17B10 Q99714 1/20 0.33
EGFR P00533 1/20 0.31
PARP1 P09874 1/20 0.31
TNKS2 Q9H2K2 1/20 0.31
PARP2 Q9UGN5 1/20 0.31
PARP3 Q9Y6F1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6092177 0.85 KDR (0.60) KDRPDGFRBFGFR1SRCRET
SCHEMBL6092180 0.85 KDR (0.60) KDRPDGFRBFGFR1SRCRET
SCHEMBL6088171 0.83 KDR (0.43) KDRPDGFRBFGFR1SRCPKN1
SCHEMBL6090570 0.81 KDR (0.43) KDRPDGFRBFGFR1SRCPKN1
SCHEMBL6090793 0.81 KDR (0.46) KDRPDGFRBFGFR1SRCPKN1
SCHEMBL6091305 0.79 KDR (0.50) KDRPDGFRBFGFR1SRCPKN1
SCHEMBL6090489 0.79 KDR (0.43) KDRPDGFRBFGFR1SRCPKN1
SCHEMBL6091313 0.79 KDR (0.50) KDRPDGFRBFGFR1SRCPKN1
SCHEMBL6092869 0.79 KDR (0.39) KDRPDGFRBFGFR1SRCRET
SCHEMBL6092868 0.79 KDR (0.39) KDRPDGFRBFGFR1SRCRET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7060822-B1 2-pyrazolin-5-ones ABBOTT GMBH & CO. KG (DE) 2006-06-13 US disclosed