SCHEMBL6089901

SCHEMBL6089901

COc1ccc2c(c1)c(C=C1C(=O)NN=C1C1CC1)cn2C

nearest known ligand 0.62

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDR P35968 7/20 0.62
GSK3B P49841 1/20 0.56
SYK P43405 9/20 0.51
FCER2 P06734 4/20 0.51
NTRK1 P04629 3/20 0.50
NTRK3 Q16288 3/20 0.50
NTRK2 Q16620 3/20 0.50
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
USP2 O75604 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6089894 1.00 KDR (0.62) KDRGSK3BSYKFCER2NTRK1
SCHEMBL6088407 0.83 KMT2A (0.57) KDRGSK3BSYKNTRK1NTRK3
SCHEMBL6088412 0.83 KMT2A (0.57) KDRGSK3BSYKNTRK1NTRK3
SCHEMBL6088475 0.80 KDR (0.62) KDRGSK3BSYKFCER2NTRK1
SCHEMBL6088468 0.80 KDR (0.62) KDRGSK3BSYKFCER2NTRK1
SCHEMBL6090500 0.77 KDR (0.45) KDRSYKFCER2NTRK1MEN1
SCHEMBL6090495 0.77 KDR (0.45) KDRSYKFCER2NTRK1MEN1
SCHEMBL7492063 0.74 PIK3CA (0.44) MEN1KMT2A
SCHEMBL5464906 0.74 SYK (0.72) KDRGSK3BSYKFCER2NTRK1
SCHEMBL5464897 0.74 SYK (0.72) KDRGSK3BSYKFCER2NTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7060822-B1 2-pyrazolin-5-ones ABBOTT GMBH & CO. KG (DE) 2006-06-13 US disclosed