SCHEMBL6090680

SCHEMBL6090680

COC(=O)C(Cc1c(C=C2C(=O)NN=C2CCc2ccc(O)cc2)[nH]c2ccccc12)NC(C)=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 4/20 0.41
ESR2 Q92731 4/20 0.41
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 2/20 0.39
PKM P14618 1/20 0.39
EGFR P00533 1/20 0.38
SRC P12931 1/20 0.38
ELANE P08246 1/20 0.38
TACR1 P25103 4/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
LMNA P02545 1/20 0.35
TP53 P04637 1/20 0.35
CYP1A2 P05177 1/20 0.35
POLB P06746 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
MAPT P10636 1/20 0.35
CYP2C9 P11712 1/20 0.35
NFKB1 P19838 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6090674 1.00 ESR1 (0.41) ESR1ESR2KDM4EALDH1A1PKM
SCHEMBL6091733 0.94 KDM4E (0.44) ESR1ESR2KDM4EALDH1A1PKM
SCHEMBL6091729 0.94 KDM4E (0.44) ESR1ESR2KDM4EALDH1A1PKM
SCHEMBL6087990 0.93 KDM4E (0.38) ESR1ESR2KDM4EALDH1A1PKM
SCHEMBL6087991 0.93 KDM4E (0.38) ESR1ESR2KDM4EALDH1A1PKM
SCHEMBL7491152 0.93 ESR1 (0.38) ESR1ESR2KDM4EALDH1A1PKM
SCHEMBL7489562 0.88 KDM4E (0.36) ESR1ESR2KDM4EALDH1A1PKM
SCHEMBL6092216 0.82 EGFR (0.40) KDM4EALDH1A1PKMEGFRSRC
SCHEMBL6090463 0.82 ALDH1A1 (0.39) ESR1ESR2KDM4EALDH1A1PKM
SCHEMBL6092220 0.82 EGFR (0.40) KDM4EALDH1A1PKMEGFRSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7060822-B1 2-pyrazolin-5-ones ABBOTT GMBH & CO. KG (DE) 2006-06-13 US disclosed