SCHEMBL6091587

SCHEMBL6091587

CCN(CC)CCc1c(C)[nH]c(/C=C2/C(=O)NN=C2c2cnccn2)c1-c1ccc(OC)cc1

nearest known ligand 0.73

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDR P35968 14/20 0.73
CHEK1 O14757 1/20 0.73
PDGFRB P09619 1/20 0.34
FGFR1 P11362 1/20 0.34
ALOX5 P09917 1/20 0.33
MCHR1 Q99705 1/20 0.33
CCNB2 O95067 3/20 0.33
CDK1 P06493 3/20 0.33
CCNB1 P14635 3/20 0.33
GSK3A P49840 3/20 0.33
GSK3B P49841 3/20 0.33
CCNB3 Q8WWL7 3/20 0.33
CDK5 Q00535 2/20 0.33
CDK5R1 Q15078 2/20 0.33
CCNE1 P24864 1/20 0.33
CDK2 P24941 1/20 0.33
ZAP70 P43403 1/20 0.33
PTK2B Q14289 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6091598 1.00 KDR (0.73) KDRCHEK1PDGFRBFGFR1ALOX5
SCHEMBL6091354 0.90 KDR (0.78) KDRCHEK1PDGFRBFGFR1
SCHEMBL6091371 0.90 KDR (0.78) KDRCHEK1PDGFRBFGFR1
SCHEMBL6088270 0.89 KDR (0.84) KDRCHEK1PDGFRBFGFR1
SCHEMBL6088236 0.89 KDR (0.84) KDRCHEK1PDGFRBFGFR1
SCHEMBL6088770 0.89 KDR (0.56) KDRCHEK1PDGFRBFGFR1ALOX5
SCHEMBL6088735 0.89 KDR (0.56) KDRCHEK1PDGFRBFGFR1ALOX5
SCHEMBL6090893 0.87 KDR (0.55) KDRCHEK1PDGFRBFGFR1ALOX5
SCHEMBL6090855 0.87 KDR (0.55) KDRCHEK1PDGFRBFGFR1ALOX5
SCHEMBL6090243 0.87 KDR (0.78) KDRCHEK1PDGFRBFGFR1ZAP70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7060822-B1 2-pyrazolin-5-ones ABBOTT GMBH & CO. KG (DE) 2006-06-13 US disclosed