SCHEMBL6097133

SCHEMBL6097133

O=C(N[C@@H](Cc1ccc(-c2ccc(C(F)(F)F)cc2)cc1)C(=O)O)c1cc(-c2ccc(F)c(Cl)c2)ccc1O

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 4/20 0.51
ITGA4 P13612 4/20 0.51
KIFC1 Q9BW19 5/20 0.50
ECE1 P42892 2/20 0.49
MRGPRX4 Q96LA9 1/20 0.46
MCL1 Q07820 1/20 0.46
CDK2 P24941 1/20 0.45
ITGB7 P26010 2/20 0.45
PSMB5 P28074 1/20 0.45
PDK1 Q15118 1/20 0.44
PDK2 Q15119 1/20 0.44
PDK3 Q15120 1/20 0.44
PDK4 Q16654 1/20 0.44
TMPRSS4 Q9NRS4 1/20 0.43
ERAP1 Q9NZ08 2/20 0.43
ALB P02768 1/20 0.43
IL2 P60568 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3991301 1.00 ITGB1 (0.51) ITGB1ITGA4KIFC1ECE1MRGPRX4
SCHEMBL4829787 1.00 ITGB1 (0.51) ITGB1ITGA4KIFC1ECE1MRGPRX4
SCHEMBL3989525 1.00 ITGB1 (0.51) ITGB1ITGA4KIFC1ECE1MRGPRX4
SCHEMBL3972237 0.94 KIFC1 (0.59) ITGB1ITGA4KIFC1ECE1MRGPRX4
SCHEMBL4824086 0.94 KIFC1 (0.59) ITGB1ITGA4KIFC1ECE1MRGPRX4
SCHEMBL13986728 0.91 PSMB5 (0.46) ITGB1ITGA4KIFC1ECE1MCL1
SCHEMBL4827782 0.91 ECE1 (0.53) ITGB1ITGA4KIFC1ECE1ITGB7
SCHEMBL4827784 0.91 ECE1 (0.53) ITGB1ITGA4KIFC1ECE1ITGB7
SCHEMBL4827806 0.90 CDK2 (0.47) ITGB1ITGA4KIFC1ECE1MCL1
SCHEMBL5544392 0.90 CDK2 (0.47) ITGB1ITGA4KIFC1ECE1MCL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7122580-B2 Aryl and heteroaryl compounds and methods to modulate coagulation TRANSTECH PHARMA, INC. (US) 2006-10-17 US disclosed