SCHEMBL6102410

SCHEMBL6102410

CC(=O)Nc1ccc(-c2ccc(C(=O)N3CCc4cc(F)c(N5C[C@@H](C)N[C@@H](C)C5)cc43)cc2)c(C)c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 10/20 0.66
HTR1B P28222 10/20 0.66
PDK1 Q15118 1/20 0.42
PDK2 Q15119 1/20 0.42
PDK3 Q15120 1/20 0.42
PDK4 Q16654 1/20 0.42
ALDH1A1 P00352 1/20 0.41
HTR1A P08908 1/20 0.40
AVPR1A P37288 1/20 0.38
XIAP P98170 1/20 0.37
BIRC2 Q13490 1/20 0.37
MAPT P10636 3/20 0.37
MEN1 O00255 2/20 0.37
HTR2A P28223 2/20 0.37
MAPK1 P28482 2/20 0.37
KMT2A Q03164 2/20 0.37
TDP1 Q9NUW8 2/20 0.37
TP53 P04637 1/20 0.37
CYP1A2 P05177 1/20 0.37
CHRM2 P08172 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6101028 0.89 HTR1D (0.60) HTR1DHTR1BHTR1AXIAPBIRC2
SCHEMBL6101995 0.89 HTR1D (0.84) HTR1DHTR1BHTR1AHTR2ASLC6A4
SCHEMBL6101776 0.87 HTR1D (0.61) HTR1DHTR1BHTR1ATP53LMNA
SCHEMBL6101016 0.86 HTR1D (0.56) HTR1DHTR1BPDK1PDK2PDK3
SCHEMBL6101864 0.85 HTR1D (0.63) HTR1DHTR1BALDH1A1HTR1AXIAP
SCHEMBL6102080 0.82 HTR1D (0.59) HTR1DHTR1BHTR1AXIAPBIRC2
SCHEMBL6100069 0.81 HTR1D (0.44) HTR1DHTR1BPDK1PDK2PDK3
SCHEMBL6166896 0.81 HTR1D (0.44) HTR1DHTR1BPDK1PDK2PDK3
SCHEMBL6101634 0.80 HTR1D (0.57) HTR1DHTR1BALDH1A1HTR1AXIAP
SCHEMBL6100063 0.79 HTR1B (0.75) HTR1DHTR1BHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7109201-B2 Piperazine derivatives, their preparation and uses in therapy SMITHKLINE BEECHAM PLC (GB) 2006-09-19 US claimed