SCHEMBL6101028

SCHEMBL6101028

Cc1cc(NS(C)(=O)=O)ccc1-c1ccc(C(=O)N2CCc3cc(F)c(N4C[C@@H](C)N[C@@H](C)C4)cc32)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 10/20 0.60
HTR1B P28222 10/20 0.60
GHSR Q92847 6/20 0.41
HTR1A P08908 1/20 0.39
TRIM24 O15164 1/20 0.38
MEN1 O00255 2/20 0.37
MAPT P10636 2/20 0.37
MAPK1 P28482 2/20 0.37
KMT2A Q03164 2/20 0.37
TDP1 Q9NUW8 2/20 0.37
HTR2A P28223 2/20 0.37
TP53 P04637 1/20 0.37
CYP1A2 P05177 1/20 0.37
CHRM2 P08172 1/20 0.37
CYP3A4 P08684 1/20 0.37
CHRM5 P08912 1/20 0.37
ADRA2A P08913 1/20 0.37
CYP2D6 P10635 1/20 0.37
CHRM1 P11229 1/20 0.37
CYP2C9 P11712 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6100097 0.89 HTR1D (0.76) HTR1DHTR1BGHSRHTR1AHTR2A
SCHEMBL6102410 0.89 HTR1D (0.66) HTR1DHTR1BHTR1AMEN1MAPT
SCHEMBL6102054 0.86 HTR1D (0.55) HTR1DHTR1BGHSRHTR1AMAPT
SCHEMBL6102080 0.85 HTR1D (0.59) HTR1DHTR1BGHSRHTR1AMEN1
SCHEMBL6101776 0.82 HTR1D (0.61) HTR1DHTR1BHTR1ATP53LMNA
SCHEMBL6101864 0.82 HTR1D (0.63) HTR1DHTR1BHTR1AMEN1MAPT
SCHEMBL6100571 0.81 GHSR (0.41) HTR1DHTR1BGHSR
SCHEMBL6099612 0.81 HTR1D (0.55) HTR1DHTR1BGHSRHTR1AMEN1
SCHEMBL6101995 0.78 HTR1D (0.84) HTR1DHTR1BGHSRHTR1AHTR2A
SCHEMBL6101016 0.78 HTR1D (0.56) HTR1DHTR1BHTR1AMEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7109201-B2 Piperazine derivatives, their preparation and uses in therapy SMITHKLINE BEECHAM PLC (GB) 2006-09-19 US claimed