SCHEMBL6108554

SCHEMBL6108554

CCCCOc1c(CN(C(=O)O)C(C)(C)C)n(CC2CC2)c(=O)c2ccc(OCC(N)=O)cc12

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 7/20 0.41
PLA2G2A P14555 3/20 0.36
AVPR1B P47901 3/20 0.34
KDM4E B2RXH2 2/20 0.34
ALDH1A1 P00352 2/20 0.34
HSD17B10 Q99714 2/20 0.34
HPGD P15428 1/20 0.34
ALOX5AP P20292 1/20 0.34
IRAK4 Q9NWZ3 1/20 0.33
ADORA2A P29274 1/20 0.33
ADORA2B P29275 1/20 0.33
ADORA1 P30542 1/20 0.33
CYP2C9 P11712 1/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6108742 0.88 AVPR1B (0.37) AVPR1BKDM4EALDH1A1SMN1; SMN2MEN1
SCHEMBL6109274 0.88 DPP4 (0.54) DPP4KDM4EALDH1A1HSD17B10HPGD
SCHEMBL6109990 0.88 GSK3B (0.35) DPP4AVPR1BKDM4EALDH1A1HSD17B10
SCHEMBL6109713 0.87 MAPK8 (0.42) DPP4AVPR1BKDM4EALDH1A1HSD17B10
SCHEMBL6108298 0.86 PGR (0.37) AVPR1BKDM4EALDH1A1HSD17B10HPGD
SCHEMBL6109025 0.85 GSK3B (0.32) AVPR1B
Hydrochloric Acid SCHEMBL5231925 0.85 DPP4 (0.51) DPP4PLA2G2AAVPR1BKDM4EALDH1A1
SCHEMBL6109704 0.84 KDM4E (0.31) AVPR1BKDM4EALDH1A1HSD17B10HPGD
SCHEMBL6109443 0.84 PARP15 (0.36) AVPR1B
SCHEMBL5235599 0.83 DPP4 (0.43) DPP4PLA2G2AAVPR1BKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7034039-B2 Fused heterocyclic compounds TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2006-04-25 US disclosed