SCHEMBL6109456

SCHEMBL6109456

COc1cc(NC(=O)Nc2ccccc2)ccc1C(=O)NCCCN1CCOCC1

nearest known ligand 0.85

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 6/20 0.85
MCHR2 Q969V1 2/20 0.73
ALDH1A1 P00352 1/20 0.66
LMNA P02545 3/20 0.65
MAPT P10636 2/20 0.61
EPHX2 P34913 5/20 0.60
PKM P14618 1/20 0.60
CYP2D6 P10635 1/20 0.57
CYP2C9 P11712 1/20 0.57
SMN1; SMN2 Q16637 1/20 0.56
TSHR P16473 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6109038 0.94 MCHR1 (0.90) MCHR1MCHR2ALDH1A1LMNAMAPT
SCHEMBL6109229 0.93 MCHR1 (0.77) MCHR1MCHR2ALDH1A1LMNAMAPT
SCHEMBL6109146 0.92 MCHR1 (1.00) MCHR1MCHR2ALDH1A1LMNAMAPT
SCHEMBL6108922 0.92 MCHR1 (0.73) MCHR1MCHR2ALDH1A1LMNAEPHX2
SCHEMBL6109418 0.91 MCHR1 (0.93) MCHR1MCHR2ALDH1A1LMNA
SCHEMBL6109289 0.91 MCHR1 (0.77) MCHR1MCHR2ALDH1A1LMNAMAPT
SCHEMBL6109770 0.91 MCHR1 (0.77) MCHR1MCHR2ALDH1A1LMNAMAPT
SCHEMBL6110331 0.88 MCHR1 (0.81) MCHR1MCHR2ALDH1A1LMNAEPHX2
SCHEMBL6109186 0.88 MCHR1 (0.70) MCHR1MCHR2ALDH1A1LMNAMAPT
SCHEMBL6110505 0.88 MCHR1 (1.00) MCHR1MCHR2ALDH1A1MAPTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060235035-A1 Novel methoxybenzamibe compounds for use in mch receptor related disorders 7TM PHARMA A/S (DK) 2006-10-19 US disclosed
WO-2004048319-A1 NOVEL BENZAMIDE COMPOUNDS FOR USE IN MCH RECEPTOR RELATED DISORDERS 7TM PHARMA A/S (DK) 2004-06-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060235035-A1 Novel methoxybenzamibe compounds for use in mch receptor related disorders GPR119, MCHR2, HCRTR2 MCHR1 5/4885MCHR2 2/4885ALDH1A1 3618/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.