Bicarbonate

Bicarbonate

SCHEMBL6130587

Cl.O=C(O)O.O=S(=O)(O)c1ccccc1C=Cc1ccccc1

nearest known ligand 0.47

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Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 2/20 0.47
NFE2L2 Q16236 3/20 0.43
HDAC1 Q13547 3/20 0.41
LMNA P02545 2/20 0.41
HDAC3 O15379 2/20 0.41
HDAC4 P56524 2/20 0.41
HDAC2 Q92769 2/20 0.41
HDAC8 Q9BY41 2/20 0.41
HDAC6 Q9UBN7 2/20 0.41
TNKS O95271 1/20 0.41
HCAR2 Q8TDS4 1/20 0.41
HDAC7 Q8WUI4 1/20 0.41
HDAC10 Q969S8 1/20 0.41
HDAC11 Q96DB2 1/20 0.41
TNKS2 Q9H2K2 1/20 0.41
HDAC9 Q9UKV0 1/20 0.41
HDAC5 Q9UQL6 1/20 0.41
PLIN1 O60240 1/20 0.41
ALDH1A1 P00352 1/20 0.41
CYP1A2 P05177 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1557243 0.95 TRPA1 (0.52) TRPA1NFE2L2HDAC1LMNAHDAC3
SCHEMBL11882514 0.95 TRPA1 (0.52) TRPA1NFE2L2HDAC1LMNAHDAC3
SCHEMBL29725577 0.95 TRPA1 (0.52) TRPA1NFE2L2HDAC1LMNAHDAC3
SCHEMBL4207529 0.95 TRPA1 (0.52) TRPA1NFE2L2HDAC1LMNAHDAC3
SCHEMBL28019442 0.93 TRPA1 (0.50) TRPA1NFE2L2HDAC1LMNAHDAC3
Ammonia Solution, Strong SCHEMBL27722454 0.93 TRPA1 (0.50) TRPA1NFE2L2HDAC1LMNAHDAC3
SCHEMBL9162326 0.89 TRPA1 (0.44) TRPA1NFE2L2CYP2D6TDP1
SCHEMBL14417984 0.88 TRPA1 (0.46) TRPA1NFE2L2HDAC1LMNAHDAC2
SCHEMBL2754803 0.88 TRPA1 (0.46) TRPA1NFE2L2HDAC1LMNAHDAC2
Isothiocyanate SCHEMBL9212863 0.85 TRPA1 (0.43) TRPA1NFE2L2LMNATDP1PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1450810-A4 XANTHINE OXIDASE INHIBITION UAB RESEARCH FOUNDATION (US) 2005-11-30 EP disclosed
EP-1450810-A2 XANTHINE OXIDASE INHIBITION THE UAB RESEARCH FOUNDATION (US) 2004-09-01 EP disclosed
US-20030158213-A1 Xanthine oxidase inhibition as a strategy to alleviate oxidative impairment of vascular function THE UAB RESEARCH FOUNDATION 2003-08-21 US disclosed
WO-2003043573-A2 XANTHINE OXIDASE INHIBITION THE UAB RESEARCH FOUNDATION (US) 2003-05-30 WO disclosed