SCHEMBL6132006

SCHEMBL6132006

COC1(OCCO)CCN(Cc2ccccc2)C1

nearest known ligand 0.50

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 5/20 0.46
TSHR P16473 3/20 0.46
CYP3A4 P08684 3/20 0.46
ALDH1A1 P00352 1/20 0.44
OPRL1 P41146 1/20 0.43
KMT2A Q03164 2/20 0.43
KDM4E B2RXH2 1/20 0.43
POLB P06746 1/20 0.43
HSD17B10 Q99714 1/20 0.42
SIGMAR1 Q99720 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20571573 0.80 CYP3A4 (0.59) CYP2D6TSHRCYP3A4ALDH1A1OPRL1
SCHEMBL11690706 0.78 OPRL1 (0.51) CYP2D6TSHRCYP3A4ALDH1A1OPRL1
SCHEMBL28447051 0.76 GAA (0.56) CYP2D6TSHRCYP3A4KMT2APOLB
SCHEMBL11686069 0.76 OPRL1 (0.52) CYP2D6TSHRCYP3A4ALDH1A1OPRL1
SCHEMBL9177696 0.75 OPRL1 (0.51) CYP2D6TSHRCYP3A4ALDH1A1OPRL1
SCHEMBL7511281 0.74 OPRL1 (0.57) CYP2D6TSHRCYP3A4ALDH1A1OPRL1
SCHEMBL11683058 0.74 OPRL1 (0.50) CYP2D6TSHRCYP3A4ALDH1A1OPRL1
Hydrochloric Acid SCHEMBL6543173 0.73 POLB (0.58) CYP2D6TSHRCYP3A4ALDH1A1OPRL1
SCHEMBL4502776 0.73 POLB (0.52) CYP2D6TSHRCYP3A4ALDH1A1KMT2A
SCHEMBL12406526 0.73 CYP3A4 (0.50) CYP2D6TSHRCYP3A4ALDH1A1OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1032559-A4 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMA INC (US) 2005-05-25 EP disclosed
US-6479495-B1 SIMULTANEOUSLY TREATING DEPRESSION AND MEMORY DYSFUNCTION IN MAMMALS SUFFERING FROM MEMORY DYSFUNCTION AND DEPRESSION AVENTIS PHARMACEUTICALS INC. 2002-11-12 US disclosed
EP-1032559-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 2000-09-06 EP disclosed
WO-1999016746-A1 AMINOALKYLPHENOL DERIVATIVES AND RELATED COMPOUNDS AVENTIS PHARMACEUTICALS INC. (US) 1999-04-08 WO disclosed