SCHEMBL6134476

SCHEMBL6134476

Nc1ncc(-c2ccc(=O)[nH]n2)c(-c2ccccc2Br)n1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.40
CLK1 P49759 9/20 0.39
CDK5 Q00535 5/20 0.39
CDK5R1 Q15078 5/20 0.39
AKR1B1 P15121 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
POLB P06746 1/20 0.36
DCUN1D1 Q96GG9 1/20 0.36
IDO1 P14902 1/20 0.35
FGFR1 P11362 1/20 0.35
CDC7 O00311 1/20 0.35
HSD17B10 Q99714 1/20 0.35
ADORA2A P29274 2/20 0.35
ADORA1 P30542 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6133466 0.85 ADORA2A (0.41) CYP1A2CLK1KDM4EALDH1A1POLB
SCHEMBL6133302 0.83 CYP1A2 (0.54) CYP1A2ADORA2AADORA1
SCHEMBL6134067 0.82 ADORA2A (0.49) ALDH1A1DCUN1D1HSD17B10ADORA2AADORA1
SCHEMBL6133777 0.81 ADORA1 (0.41) CYP1A2CLK1AKR1B1ADORA2AADORA1
SCHEMBL6134475 0.80 ADORA1 (0.41) CYP1A2CLK1CDK5CDK5R1ALDH1A1
SCHEMBL11633235 0.79 CYP1A2 (0.56) CYP1A2AKR1B1KDM4EPOLBDCUN1D1
SCHEMBL6134600 0.79 FGFR1 (0.42) CYP1A2CLK1CDK5CDK5R1POLB
SCHEMBL6133799 0.78 ADORA2A (0.54) CDK5CDK5R1KDM4EALDH1A1POLB
SCHEMBL6133893 0.78 FGFR1 (0.43) CYP1A2AKR1B1FGFR1ADORA2AADORA1
SCHEMBL6133404 0.78 CYP1A2 (0.37) CYP1A2CLK1CDK5CDK5R1AKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050043315-A1 Aminopyrimidine compounds, processes for their preparation and pharmaceutical compositions containing them ASTELLAS PHARMA INC. (JP) 2005-02-24 US disclosed
WO-2003057689-A1 AMINOPYRIMIDINE COMPOUNDS, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-07-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050043315-A1 Aminopyrimidine compounds, processes for their preparation and pharmaceutical compositions containing them ADORA2B, ADORA2A, ADORA1 CYP1A2 1170/4885CLK1 3624/4885CDK5 823/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.