SCHEMBL6135055

SCHEMBL6135055

COC(=O)c1ccc(C(=O)NNC(=O)c2ccc(OC3CCN(c4ccccc4)CC3)cc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACACB O00763 1/20 0.49
NPC1 O15118 3/20 0.48
RAB9A P51151 2/20 0.48
KMT2A Q03164 3/20 0.48
NAMPT P43490 1/20 0.47
TSHR P16473 1/20 0.47
HTT P42858 1/20 0.47
MAPT P10636 3/20 0.47
MEN1 O00255 2/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
HPGD P15428 1/20 0.47
FFAR4 Q5NUL3 1/20 0.47
HRH3 Q9Y5N1 1/20 0.46
SRD5A1 P18405 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
LMNA P02545 2/20 0.46
OPRM1 P35372 1/20 0.46
OPRD1 P41143 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6135625 0.91 ALDH1A1 (0.52) ACACBNPC1RAB9AKMT2AHTT
SCHEMBL6135560 0.83 FFAR4 (0.53) ACACBNPC1RAB9AKMT2ANAMPT
SCHEMBL6134747 0.83 NPC1 (0.48) ACACBNPC1RAB9AKMT2ANAMPT
SCHEMBL6135447 0.81 ALDH1A1 (0.55) ACACBKMT2ANAMPTTSHRMAPT
SCHEMBL31162683 0.79 FFAR4 (0.50) ACACBNAMPTMAPTFFAR4HDAC8
SCHEMBL6135385 0.79 HRH3 (0.60) KMT2AMEN1HRH3
Acetic Acid Methyl Ester SCHEMBL31162636 0.79 FFAR4 (0.55) ACACBKMT2ANAMPTMEN1HPGD
SCHEMBL31162733 0.78 FFAR4 (0.59) ACACBKMT2ANAMPTMAPTMEN1
SCHEMBL22694560 0.77 KMT2A (0.51) KMT2AMEN1HRH3SRD5A1LMNA
SCHEMBL6133632 0.77 HDAC3 (0.48) NPC1RAB9ATSHRMAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050261177-A1 Compound ASTELLAS PHARMA INC. (JP) 2005-11-24 US disclosed
EP-1366066-A2 CYCLOHEXAPEPTIDE HAVING ANTIMICROBIAL ACTIVITY FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-12-03 EP disclosed
WO-2002072621-A2 CYCLOHEXAPEPTIDE HAVING ANTIMICROBIAL ACTIVITY FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-09-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050261177-A1 Compound MANBA, MAN2B1, MAN2A1 ACACB 4561/4885NPC1 1070/4885RAB9A 3326/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.