SCHEMBL6135652

SCHEMBL6135652

Fc1cc(-n2nnc(-c3ccccn3)n2)ccc1-c1ccccn1.N#Cc1cc(-n2nnc(-c3ccccn3)n2)ccc1-c1ccccn1

nearest known ligand 0.68

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 10/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3371658 0.93 GRM5 (0.67) GRM5
SCHEMBL3371020 0.90 GRM5 (0.65) GRM5
SCHEMBL4700139 0.88 GRM5 (0.65) GRM5
SCHEMBL13684154 0.84 GRM5 (0.60) GRM5
SCHEMBL4699537 0.81 GRM5 (0.65) GRM5
SCHEMBL4701864 0.80 GRM5 (0.67) GRM5
SCHEMBL4698815 0.79 GRM5 (0.65) GRM5
SCHEMBL4703812 0.77 GRM5 (0.63) GRM5
SCHEMBL4699189 0.77 GRM5 (0.65) GRM5
SCHEMBL13683937 0.76 GRM5 (0.61) GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1485093-A4 DI-ARYL SUBSTITUTED TETRAZOLE MODULATORS OF METABOTROPIC GLUTAMATE RECEPTOR-5 MERCK & CO INC (US) 2005-12-28 EP disclosed
EP-1485093-A1 DI-ARYL SUBSTITUTED TETRAZOLE MODULATORS OF METABOTROPIC GLUTAMATE RECEPTOR-5 Merck & Co., Inc. (US) 2004-12-15 EP disclosed
WO-2003077918-A1 DI-ARYL SUBSTITUTED TETRAZOLE MODULATORS OF METABOTROPIC GLUTAMATE RECEPTOR-5 MERCK & CO., INC. (US) 2003-09-25 WO disclosed