SCHEMBL6141402

SCHEMBL6141402

C[C@]1(C(=O)[AsH][C@@H](Cc2ccc3nc(-c4c(Cl)cccc4Cl)ccc3c2)C(=O)O)CCCO1

nearest known ligand 0.50

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 18/20 0.50
ITGAV P06756 1/20 0.50
ITGA4 P13612 17/20 0.37
ITGB7 P26010 6/20 0.37
ABL1 P00519 1/20 0.36
KCNH2 Q12809 1/20 0.32
HRH3 Q9Y5N1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6141406 1.00 ITGB1 (0.50) ITGB1ITGAVITGA4ITGB7ABL1
SCHEMBL3312652 0.84 ITGB1 (0.65) ITGB1ITGAVITGA4ITGB7
SCHEMBL3312661 0.84 ITGB1 (0.65) ITGB1ITGAVITGA4ITGB7
SCHEMBL4625549 0.80 ITGB1 (0.54) ITGB1ITGAVITGA4ITGB7ABL1
SCHEMBL6142370 0.78 ITGB1 (0.66) ITGB1ITGAVITGA4ITGB7ABL1
SCHEMBL6141473 0.77 ITGB1 (0.55) ITGB1ITGAVITGA4ITGB7ABL1
SCHEMBL3312918 0.77 ITGB1 (0.62) ITGB1ITGAVITGA4ITGB7
SCHEMBL3312924 0.77 ITGB1 (0.62) ITGB1ITGAVITGA4ITGB7
SCHEMBL6141061 0.76 ITGB1 (0.55) ITGB1ITGAVITGA4ITGB7ABL1
SCHEMBL6141563 0.76 ITGB1 (0.46) ITGB1ITGAVITGA4ITGB7ABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501801-A1 2,6-QUINOLINYL AND 2,6-NAPHTHYL DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES AS VLA-4 INHIBITORS UCB, S.A. (BE) 2005-02-02 EP disclosed
WO-2003093237-A1 2,6-QUINOLINYL AND 2,6-NAPHTHYL DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES AS VLA-4 INHIBITORS UCB, S.A. (BE) 2003-11-13 WO disclosed